Last update 25 Jul 2026

CP-161242

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
CP-161242
Target
5-HT1D receptor
Action
partial agonists
Mechanism
5-HT1D receptor partial agonists(Serotonin 1d (5-HT1d) receptor partial agonists)
Therapeutic Areas
Nervous System DiseasesOther Diseases
Active Indication-
Inactive Indication
Anxiety DisordersDepressive DisorderMigraine Disorders
Originator Organization
Pfizer Inc.Pfizer Inc.
Active Organization-
Inactive Organization
Pfizer Inc.Pfizer Inc.
License Organization-
Drug Highest PhasePendingDiscovery
First Approval Date-
Regulation-

Structure/Sequence

Molecular FormulaC22H21N5
InChIKeyKVKYGVOAHGNAKZ-QGZVFWFLSA-N
CAS Registry160906-61-6

Related

100 Clinical Results associated with CP-161242
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100 Translational Medicine associated with CP-161242
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100 Patents (Medical) associated with CP-161242
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2
Literatures (Medical) associated with CP-161242
01 Oct 1995BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
5-cyano-1-[3-(N-methylpyrrolidin-2R-ylmethyl)indol-5-yl] benzimidazole (CP-161,242): A potent, centrally active 5-HT1D receptor agonist and benzodiazepine partial agonist
01 Oct 1995BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
The discovery of a novel and potent benzodiazepine receptor pharmacophore
100 Deals associated with CP-161242
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R&D Status

10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
Anxiety DisordersDiscovery
United States
Pfizer Inc.Pfizer Inc.
-
Depressive DisorderDiscovery
United States
Pfizer Inc.Pfizer Inc.
-
Migraine DisordersDiscovery
United States
Pfizer Inc.Pfizer Inc.
-
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date

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Clinical Trial

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Approval

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Regulation

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