Drug Type Small molecule drug |
Synonyms W 4032, W4032 |
Target |
Action inhibitors |
Mechanism EHMT2 inhibitors(euchromatic histone lysine methyltransferase 2 inhibitors), NSD2 inhibitors(nuclear receptor binding SET domain protein 2 inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication- |
Originator Organization |
Active Organization |
Inactive Organization- |
License Organization- |
Drug Highest PhasePreclinical |
First Approval Date- |
Regulation- |
Molecular FormulaC25H36N6O2 |
InChIKeyKKXRBRPMTQSNTJ-UHFFFAOYSA-N |
CAS Registry2761292-51-5 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Neoplasms | Preclinical | China | 15 Jul 2024 |