Last update 30 Apr 2026

Bezafibrate/Diflunisal

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
bezafibrate + diflunisal, Diflunisal/bezafibrate, CRX-401
Target
COXs x PPARα
Action
inhibitors, agonists
Mechanism
COX inhibitors(Cyclooxygenases inhibitors), PPARα agonists(Peroxisome proliferator-activated receptor α agonists)
Therapeutic Areas
Endocrinology and Metabolic Disease
Active Indication-
Inactive Indication
Diabetes Mellitus, Type 2
Originator Organization
Zalicus, Inc.Zalicus, Inc.
Active Organization-
Inactive Organization
Zalicus, Inc.Zalicus, Inc.
License Organization-
Drug Highest PhaseDiscontinuedPhase 2
First Approval Date-
Regulation-
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Structure/Sequence

Molecular FormulaC13H8F2O3
InChIKeyHUPFGZXOMWLGNK-UHFFFAOYSA-N
CAS Registry22494-42-4
View All Structures (2)

Related

1
Clinical Trials associated with Bezafibrate/Diflunisal
NCT00506298
/ CompletedPhase 2
A Randomized, Multi-Center Study to Compare the Effects of CRx-401 to Bezafibrate Plus Placebo on Plasma Glucose Levels When Given to Subjects With Type II Diabetes on Metformin.
100 Clinical Results associated with Bezafibrate/Diflunisal
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100 Translational Medicine associated with Bezafibrate/Diflunisal
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100 Patents (Medical) associated with Bezafibrate/Diflunisal
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100 Deals associated with Bezafibrate/Diflunisal
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External Link

KEGGWikiATCDrug Bank
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DB05775

R&D Status

10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
Diabetes Mellitus, Type 2Phase 2
Canada
Zalicus, Inc.Zalicus, Inc.
01 Jul 2007
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
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Approval

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Regulation

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