Drug Type Proteolysis-targeting chimeras (PROTAC) |
Synonyms- |
Action inhibitors, degraders |
Mechanism ERK1 inhibitors(Extracellular-signal-regulated kinase1 inhibitors), FLT3 degraders(Tyrosine-protein kinase receptor FLT3 degraders), IKKα inhibitors(component of inhibitor of nuclear factor kappa B kinase complex inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication- |
Originator Organization |
Active Organization |
Inactive Organization- |
License Organization- |
Drug Highest PhasePreclinical |
First Approval Date- |
Regulation- |
| Indication | Highest Phase | Country/Location | Organization | Date |
|---|---|---|---|---|
| Acute Myeloid Leukemia | Preclinical | United States | 03 Nov 2025 | |
| B-Cell Leukemia | Preclinical | United States | 03 Nov 2025 | |
| Myelofibrosis | Preclinical | United States | 03 Nov 2025 |





