Drug Type Proteolysis-targeting chimeras (PROTAC) |
Synonyms- |
Target |
Action degraders, inhibitors |
Mechanism BRD4 degraders(Bromodomain-containing protein 4 degraders), BRD7 inhibitors(Bromodomain-containing protein 7 inhibitors), BRD9 inhibitors(Bromodomain-containing protein 9 inhibitors) |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
Inactive Organization |
License Organization- |
Drug Highest PhasePendingPreclinical |
First Approval Date- |
Regulation- |
Molecular FormulaC44H53N7O9S2 |
InChIKeyWPBRCJAGSVKMMS-UHFFFAOYSA-N |
CAS Registry2097509-20-9 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Neoplasms | Preclinical | United States | 18 Apr 2017 |