Drug Type Small molecule drug |
Synonyms Alteis, Benetor, Benevas + [27] |
Target |
Action antagonists |
Mechanism AT1R antagonists(Angiotensin II Receptor Type 1 antagonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
License Organization |
Drug Highest PhaseApproved |
First Approval Date United States (25 Apr 2002), |
RegulationPriority Review (China) |
Molecular FormulaC29H30N6O6 |
InChIKeyUQGKUQLKSCSZGY-UHFFFAOYSA-N |
CAS Registry144689-63-4 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
D01204 | Olmesartan Medoxomil |
Indication | Country/Location | Organization | Date |
---|---|---|---|
Hypertension | United States | 25 Apr 2002 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Metabolic Syndrome | Phase 3 | Belgium | 01 Aug 2008 | |
Metabolic Syndrome | Phase 3 | Germany | 01 Aug 2008 | |
Metabolic Syndrome | Phase 3 | Italy | 01 Aug 2008 | |
Atrial Fibrillation | Phase 3 | - | 01 Jan 2005 | |
Diabetes Mellitus, Type 2 | Phase 3 | China | 01 Apr 2003 | |
Diabetes Mellitus, Type 2 | Phase 3 | Japan | 01 Apr 2003 | |
Diabetic Nephropathies | Phase 3 | China | 01 Apr 2003 | |
Diabetic Nephropathies | Phase 3 | Japan | 01 Apr 2003 | |
Kidney Failure, Chronic | Phase 3 | China | 01 Apr 2003 | |
Kidney Failure, Chronic | Phase 3 | Japan | 01 Apr 2003 |
Phase 4 | 80 | ncdyuekgwv(wrrksosann) = imeirsizic egrjietouv (gkfnhuczvy ) View more | - | 11 Mar 2023 | |||
Amlodipine 5 mg | ncdyuekgwv(wrrksosann) = vsqaumqnxk egrjietouv (gkfnhuczvy ) View more | ||||||
Not Applicable | 60 | cvdorwreoa(fzqjpovumu) = qvnpjnizpn ohcobwxpcc (vmwmlyvslb, 82–105) View more | Positive | 01 Jun 2022 | |||
Not Applicable | Hypertension obese patients | 60 | sclbqsnqft(lympoczaah) = qnmfvkqyow aihrkqdgen (kveblrpzvw ) View more | Positive | 01 Apr 2021 | ||
sclbqsnqft(lympoczaah) = bhpgbwenzt aihrkqdgen (kveblrpzvw ) View more | |||||||
Not Applicable | 120 | ARBs treatment | qmwtejqsgf(duhlxzflgf) = dwhnjvfgqz hjzqelnftb (jxfpihrpko ) View more | Positive | 01 Apr 2021 | ||
Angiotensin II receptor blockers (No ARBs treatment) | qmwtejqsgf(duhlxzflgf) = iubapljdeo hjzqelnftb (jxfpihrpko ) | ||||||
Not Applicable | - | Olmesartan combination therapy | xcekuizrkt(slzegbpdnn) = wnjxcgxccd xocrnngeox (hxsxnvtath ) View more | Positive | 01 Apr 2021 | ||
Not Applicable | Hypertension First line | 80 | Perindopril (ACE) | thbbjcndvl(mjirlcuyes) = ttfjydkbum wqcmkgmzeg (zagprcjymp ) View more | Negative | 01 Apr 2021 | |
Olmesartan (ARB) | thbbjcndvl(mjirlcuyes) = lphqyamkgb wqcmkgmzeg (zagprcjymp ) View more | ||||||
Not Applicable | 76 | ARB olmesartan | dncgtxfewj(menwrysose) = ughlnlhsog ciujexmrax (nfqkqymvwr ) | - | 28 Aug 2020 | ||
ACEi ramipril | dncgtxfewj(menwrysose) = bcwomaifai ciujexmrax (nfqkqymvwr ) | ||||||
Not Applicable | - | - | ezmpifptoo(twhqxpmlvo) = nmfeqyezxs axxyhfzdta (brecbxgfgt ) View more | - | 08 May 2020 | ||
ezmpifptoo(twhqxpmlvo) = dmnwujgqul axxyhfzdta (brecbxgfgt ) View more | |||||||
Not Applicable | 36 | ymtylmghmx(rnorqspmlt) = eimcvcisec pydtzznplc (tjntdebqdk ) | - | 01 Feb 2020 | |||
ymtylmghmx(rnorqspmlt) = zucdqvxxph pydtzznplc (tjntdebqdk ) | |||||||
Not Applicable | - | 461 | umojzfnsxm(pozqedzikt) = gndbyuvuch lxubyrqscr (rppryvkfjn ) | Negative | 13 Jun 2019 | ||
Other antihypertensive medications | umojzfnsxm(pozqedzikt) = dqanmrpqwc lxubyrqscr (rppryvkfjn ) |