Drug Type Small molecule drug |
Synonyms OP 3136 |
Target |
Action inhibitors |
Mechanism KAT6A inhibitors(lysine acetyltransferase 6A inhibitors), KAT6B inhibitors(lysine acetyltransferase 6B inhibitors), Epigenetic drug |
Therapeutic Areas |
Inactive Indication- |
Originator Organization |
Active Organization |
Inactive Organization- |
License Organization |
Drug Highest PhasePhase 1 |
First Approval Date- |
Regulation- |
Molecular FormulaC20H22N4O7S |
InChIKeyKZSVPOQXJZQAQQ-UHFFFAOYSA-N |
CAS Registry3056105-63-3 |
| Indication | Highest Phase | Country/Location | Organization | Date |
|---|---|---|---|---|
| ER-positive/HER2-negative Breast Cancer | Phase 1 | United States | 16 Dec 2024 | |
| ER-positive/HER2-negative Breast Cancer | Phase 1 | Australia | 16 Dec 2024 | |
| ER-positive/HER2-negative Breast Cancer | Phase 1 | France | 16 Dec 2024 | |
| ER-positive/HER2-negative Breast Cancer | Phase 1 | Hong Kong | 16 Dec 2024 | |
| ER-positive/HER2-negative Breast Cancer | Phase 1 | Ireland | 16 Dec 2024 | |
| ER-positive/HER2-negative Breast Cancer | Phase 1 | Spain | 16 Dec 2024 | |
| Metastatic breast cancer | Phase 1 | United States | 16 Dec 2024 | |
| Metastatic breast cancer | Phase 1 | Australia | 16 Dec 2024 | |
| Metastatic breast cancer | Phase 1 | France | 16 Dec 2024 | |
| Metastatic breast cancer | Phase 1 | Hong Kong | 16 Dec 2024 |
Phase 1 | 32 | nkzsiittoe(tzqtqatuuf) = No dose-limiting toxicities (DLTs) zfpzkjapgv (grzshtoqob ) View more | Positive | 29 May 2026 | |||
Phase 1 | - | msoteqbymr(icwadjdnuu) = rblgrlupbb qesmfebpgy (lbzchidlwx ) | Positive | 28 Apr 2025 | |||
msoteqbymr(icwadjdnuu) = fbyecspffg qesmfebpgy (lbzchidlwx ) |





