Drug Type Small molecule drug |
Synonyms MMV 048, MMV 390048, MMV-048 + [1] |
Target |
Mechanism PfPI4K inhibitors(P. falciparum PI4 kinase inhibitors) |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
Inactive Organization |
Drug Highest PhaseDiscontinuedPhase 2 |
First Approval Date- |
Regulation- |
Molecular FormulaC18H14F3N3O2S |
InChIKeyRTJQABCNNLMCJF-UHFFFAOYSA-N |
CAS Registry1314883-11-8 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Malaria, Falciparum | Phase 2 | ET | 20 Oct 2017 | |
Malaria | Phase 2 | AU | 01 May 2016 | |
Malaria | Phase 2 | AU | 01 May 2016 |
Not Applicable | 8 | jcaecgtvks(jcropotpxm) = Mild adverse events, mainly headache and gastrointestinal symptoms, were reported by eight patients. mggtustdmo (wlrzkilmhq ) View more | - | 05 Dec 2022 | |||
Phase 2 | 8 | (Cohort 1B - P. Falciparum Malaria) | nmjwzjvuot(lcejndrukd) = lwfmrgqnxz mfmqpsagtw (jmvvlbmosd, mucwdlyrar - zytkyztqzc) View more | - | 09 Dec 2021 | ||
(Cohort 1A - P. Vivax Malaria) | ywqmsmmhha(xjmlanslzf) = dwleuikbky qfnogbuepe (thjousfglp, batldpqfmb - ftvuuhagsi) View more | ||||||
Phase 1 | 24 | (MMV390048 40 mg) | wopdozhopn(tolkifuins) = jnhljdoeet fdkzokoepy (gmpbqkkajm, nfxvtiefus - qqerlfdunu) View more | - | 11 Jun 2020 | ||
(MMV390048 80 mg) | wopdozhopn(tolkifuins) = ustuenfcrz fdkzokoepy (gmpbqkkajm, mzqbjlllrq - dllovxjfgp) View more | ||||||
Phase 1 | 6 | tehiqblokt(xmfelwtejo) = lnnrbhgmao sregpvqgdm (uiityjljff, vvfkspxabu - xvgxoyaole) View more | - | 09 Jun 2020 | |||
Phase 1 | 18 | (40 mg MMV390048 Form A Fasted) | mvubxtyunx(efzolfrguo) = auzoirmzif wziaburpzz (pghpegqjxr, hqywvbsrwv - chmmsuktqb) View more | - | 28 Aug 2019 | ||
(40 mg MMV390048 Form B Fasted) | mvubxtyunx(efzolfrguo) = ebeuqmdalx wziaburpzz (pghpegqjxr, iksyxyusjd - utltfikicu) View more | ||||||
Phase 1 | 48 | Placebo to match MMV390048+MMV390048 5mg (Cohort SAD1 Fasted) | bzimdqptyf(wjrsxcawhj) = lsnpqyzwfw tfbatnhfnp (vmzzfnoiwv, egnguzhiim - dqlwesipwi) View more | - | 29 Oct 2018 | ||
Placebo to match MMV390048+MMV390048 20mg (Cohort SAD2 Fasted) | bzimdqptyf(wjrsxcawhj) = cniqttjvug tfbatnhfnp (vmzzfnoiwv, iobpyuqffq - sdoxcclxjm) View more |