Last update 26 Jul 2024

Ritlecitinib Tosilate

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
Ritlecitinib, PF 06651600, PF 6651600
+ [5]
Mechanism
JAK3 inhibitors(Tyrosine-protein kinase JAK3 inhibitors), TEC inhibitors(tec protein tyrosine kinase inhibitors)
Originator Organization
Inactive Organization-
Drug Highest PhaseApproved
First Approval Date
US (23 Jun 2023),
RegulationBreakthrough Therapy (US), Priority Review (CN), Breakthrough Therapy (CN)
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Structure

Molecular FormulaC15H19N5O
InChIKeyCBRJPFGIXUFMTM-WDEREUQCSA-N
CAS Registry1792180-81-4

External Link

KEGGWikiATCDrug Bank
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R&D Status

Approved
10 top approved records.
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IndicationCountry/LocationOrganizationDate
Alopecia Areata
US
23 Jun 2023
Developing
10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
Nonsegmental vitiligoPhase 3
US
01 Dec 2022
Nonsegmental vitiligoPhase 3
CN
01 Dec 2022
Nonsegmental vitiligoPhase 3
JP
01 Dec 2022
Nonsegmental vitiligoPhase 3
AU
01 Dec 2022
Nonsegmental vitiligoPhase 3
BG
01 Dec 2022
Nonsegmental vitiligoPhase 3
CA
01 Dec 2022
Nonsegmental vitiligoPhase 3
DE
01 Dec 2022
Nonsegmental vitiligoPhase 3
IN
01 Dec 2022
Nonsegmental vitiligoPhase 3
IT
01 Dec 2022
Nonsegmental vitiligoPhase 3
MX
01 Dec 2022
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Phase 2/3
191
Ritlecitinib 50mg QD
ltwawgybbk(tbasntmwkr) = lhpkwlpngz wfvbykzdzu (qyhrsjkpwa )
-
11 Oct 2023
Phase 3
447
Ritlecitinib 200 mg
untgnvsdxc(nmwrgxrugn) = szxqnwcqok jxcdkqjzgd (xqvqutwkai )
-
11 Oct 2023
Ritlecitinib 50 mg
untgnvsdxc(nmwrgxrugn) = hldxulvevz jxcdkqjzgd (xqvqutwkai )
Phase 1
-
12
(Treatment A: Ritlecitinib 30 mg Intact Adult Capsule)
lwmkjlddta(fujrcyalhw) = sougreyhki khhzfenqge (tvrmvtvydc, xpwzulvfjt - wwdfrppzui)
-
21 Aug 2023
(Treatment B: Ritlecitinib 3*10 mg Pediatric Capsules)
lwmkjlddta(fujrcyalhw) = mitlxcwuwf khhzfenqge (tvrmvtvydc, mpgewdrlbv - evgennjdgu)
Phase 2/3
718
skbhvvxekh(dazesmzbwh) = alpeiowcfa ukfswelivg (naclcemhyl )
Positive
06 Jul 2023
skbhvvxekh(dazesmzbwh) = zbsmldlqou ukfswelivg (naclcemhyl )
Phase 3
447
tujokbpyuo(fdygksppwk) = xwjxwzsfbz ppaqhteiuy (pplelxmiym )
Positive
06 Jul 2023
fyhbidxjwg(nixlqaqadj) = phjrqlohfs kvbxpuocfl (lcwmvltnnc )
Not Applicable
261
LITFULO 50 mg QD
rvlxfqmhee(hbbxcgxplz) = Most common adverse reactions (incidence ≥1%) are headache, diarrhea, acne, rash, urticaria, folliculitis, pyrexia, atopic dermatitis, dizziness, blood creatine phosphokinase increased, herpes zoster, red blood cell count decreased, and stomatitis. uedkogjbwt (fhscxbuxqx )
Positive
23 Jun 2023
Placebo
Phase 2/3
718
oxutdclubi(kodzawukah): P-Value = 0·0002
-
13 Apr 2023
Placebo
Phase 2
460
(PF-06650833 400mg MR + Tofacitinib 11mg MR)
tvzgyqyfsm(fmnbeevror) = snwwxlsutx zwdjqboosb (inavvnotll, mvzudkohyp - rljiqjofip)
-
07 Apr 2023
(PF-06650833 400mg MR + PF-06651600 100mg)
tvzgyqyfsm(fmnbeevror) = iueykldnes zwdjqboosb (inavvnotll, uhhbvhundx - nhwwmuaycs)
Phase 2/3
-
Ritlecitinib 10 mg
acukcndagj(mttozjzimb) = touaxeciml gjdjmprerf (fyhjjmnxlb )
-
17 Mar 2023
Ritlecitinib 30 mg
acukcndagj(mttozjzimb) = jmxfsqyent gjdjmprerf (fyhjjmnxlb )
Phase 2
319
vzgvvcsbpn(mlyjostycy) = One death due to myocardial infarction (ritlecitinib) twsscstmna (zfoolugtqq )
Positive
06 Jan 2023
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