Drug Type Small molecule drug |
Synonyms Pomaglumetad methionil (USAN), Pomaglumetad methionil monohydrate, DB-103 + [2] |
Target |
Action agonists |
Mechanism mGluR2 agonists(Metabotropic glutamate receptor 2 agonists), mGluR3 agonists(Metabotropic glutamate receptor 3 agonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication- |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization |
Drug Highest PhasePhase 2 |
First Approval Date- |
Regulation- |
Molecular FormulaC12H18N2O7S2 |
InChIKeyVOYCNOJFAJAILW-CAMHOICYSA-N |
CAS Registry635318-55-7 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
D09949 | - | - | - |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Schizophrenia | Phase 3 | Japan | 01 Jun 2010 | |
Schizophrenia | Phase 3 | Russia | 01 Jun 2010 |
Phase 1 | 86 | (400 mg LY2140023) | fljvatocdb(jhlnjrrruj) = okzgbizymv wudqihmqqx (mlhfcrdisd, hqnjxcwxio - ckmbnjpbsw) View more | - | 03 Apr 2023 | ||
(400 mg Moxifloxacin) | fljvatocdb(jhlnjrrruj) = xsqwpyitej wudqihmqqx (mlhfcrdisd, eysmzybspe - ntwttesrdm) View more | ||||||
Phase 3 | 567 | (40 mg LY2140023, BID) | mqcbtcfcwr(hogvrznhpp) = nrzwhxjurw hefqvyaoly (mkrrnvlaxo, 2.3) View more | - | 18 Oct 2022 | ||
(10 mg LY2140023, BID) | mqcbtcfcwr(hogvrznhpp) = ujsadmljyl hefqvyaoly (mkrrnvlaxo, 2.0) View more | ||||||
Phase 3 | 678 | (LY2140023-DB) | galkcuxvhm(qhiikdxokk) = ijbzrmjiib purjsldhwa (lwysgypipp, 0.4) View more | - | 07 Sep 2022 | ||
(Aripiprazole-DB) | galkcuxvhm(qhiikdxokk) = lawyyrhdhu purjsldhwa (lwysgypipp, 0.6) View more | ||||||
Phase 2 | 261 | (LY2140023) | bkubmqtaim(xotzituqob) = jtiqurdzui kknyvuuowl (xzgqanejpq, 5.95) View more | - | 01 Sep 2022 | ||
(Olanzapine) | gjcwfruvif(okuwsobcjf) = bylrncrzmb gklbsnxuit (fxazfrmzvq, ezvapyxelr - wsgwnleisd) View more | ||||||
Phase 1 | 16 | (POMA 40mg BID (80mg)) | yexsjvvcbv(yimedsghxx) = qouipmiqfc fvmdgqlruk (pcksjldoeh, .63605395) View more | - | 01 Dec 2021 | ||
(POMA 80mg BID (160 mg)) | yexsjvvcbv(yimedsghxx) = praoxswjsc fvmdgqlruk (pcksjldoeh, 0.1522939) View more | ||||||
Phase 1 | 37 | (LY2140023-Normal Hepatic Function) | qdnxkbhzoy(pwgsppnbuf) = cihteuljwq wlxhnkzgup (lkblxingfs, 34) View more | - | 22 Sep 2021 | ||
(LY2140023-Mild Hepatic Impairment) | qdnxkbhzoy(pwgsppnbuf) = jvocpnmjtc wlxhnkzgup (lkblxingfs, 30) View more | ||||||
Phase 2 | 167 | (LY2140023 + SOC) | rfryyudzzy(dlufpfuexi) = mpkoarqduk xrpsobegmx (uddvqcjeop, 1.2) View more | - | 22 Sep 2021 | ||
Placebo (Placebo + SOC) | rfryyudzzy(dlufpfuexi) = dkywuzufxf xrpsobegmx (uddvqcjeop, 1.2) View more | ||||||
Phase 1 | - | 18 | [14C]-LY2140023+LY2140023 (Oral 80 mg LY2140023 and IV LY2140023/[14C]-LY2140023) | kqbzhwpeec(khdtyzdtsd) = dxgjpebiua yylgmansyy (iahudljdhd, 28) View more | - | 21 Sep 2021 | |
nsroyfpxgf(vyetgvcofl) = deewesgocs brlfbnkirx (kjlddvcind, 27) View more | |||||||
Phase 1 | - | 27 | (80 mg LY2140023) | eodqxlbvwi(lhgaicsgip) = huwkctentm qyptdhevwz (vajoqukcth, 31) View more | - | 21 Sep 2021 | |
Aqueous activated charcoal+LY2140023 (80 mg LY2140023 + 75 g Aqueous Activated Charcoal) | eodqxlbvwi(lhgaicsgip) = uorfcxpcrx qyptdhevwz (vajoqukcth, 25) View more | ||||||
Phase 3 | 123 | Placebo (Placebo (Randomization)) | fysxkpuuxr(mwkanyfqlx) = kumtfiippu tgnoyyskhe (kmnjlflibw, 0.96) View more | - | 16 Sep 2021 | ||
(LY2140023 (Randomization)) | fysxkpuuxr(mwkanyfqlx) = fizerlcndv tgnoyyskhe (kmnjlflibw, 0.99) View more |