Drug Type Synthetic peptide |
Synonyms Thymalfaxin, Thymosin alpha1 (human), Thymosin-α-1 + [8] |
Target |
Action antagonists |
Mechanism 5-HT6 receptor antagonists(Serotonin 6 (5-HT6) receptor antagonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Inactive Organization |
Drug Highest PhaseApproved |
First Approval Date China (01 Jan 1996), |
RegulationOrphan Drug (United States) |
Molecular FormulaC129H215N33O55 |
InChIKeyNZVYCXVTEHPMHE-ZSUJOUNUSA-N |
CAS Registry62304-98-7 |
Indication | Country/Location | Organization | Date |
---|---|---|---|
Hepatitis B, Chronic | China | 01 Jan 1996 | |
Hepatitis B | - | - | - |
Hepatitis C | - | - | - |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Sepsis | Phase 3 | China | 06 Sep 2016 | |
Hepatitis C, Chronic | Phase 3 | United States | 01 Apr 2002 | |
Hepatitis C, Chronic | Phase 3 | Puerto Rico | 01 Apr 2002 | |
Advanced Malignant Solid Neoplasm | Phase 2 | China | 01 Apr 2023 | |
Kidney Failure, Chronic | Phase 2 | Italy | 01 Nov 2009 | |
Hepatocellular Carcinoma | Phase 2 | United States | 28 Apr 2004 | |
Malignant melanoma, metastatic | Phase 2 | France | 01 Jul 2002 | |
Malignant melanoma, metastatic | Phase 2 | Germany | 01 Jul 2002 | |
Malignant melanoma, metastatic | Phase 2 | Hungary | 01 Jul 2002 | |
Malignant melanoma, metastatic | Phase 2 | Italy | 01 Jul 2002 |
Phase 3 | 1,106 | ivekwuiokh(hivnfjnhum) = bqpcuhtpcz hxqbtuwmay (akcogeegkr ) | Negative | 15 Jan 2025 | |||
Placebo | ivekwuiokh(hivnfjnhum) = hljmffpjcr hxqbtuwmay (akcogeegkr ) | ||||||
Phase 2 | Metastatic Solid Tumor T lymphocyte count | 6 | PRaG regimen + Thymalfasin | kjgzeqkhim(peyupiopiy) = ezouzaongh neudqojstr (eavitvcxtz ) View more | Positive | 01 Oct 2024 | |
Early Phase 1 | HIV Infections PD-1 | TIM-3 | sjTREC | 20 | Thymosin α1 1.6 mg | pckxzrpxzl(jnzrrqjznz) = qzxzvaxlyo lzhxojblis (ippgtlaqfk ) View more | Positive | 17 Jan 2024 | |
Thymosin α1ral therapy | pckxzrpxzl(jnzrrqjznz) = pgeyrmyctj lzhxojblis (ippgtlaqfk ) View more | ||||||
Phase 2 | 69 | Thymosin α1 + CCRT | cadlzqekov(jpooelkzvn) = bzxijmampo vyfwlsjnch (uhvxutlrld ) View more | Positive | 20 Jul 2022 | ||
CCRT alone | czytehxsww(smjdnfqzgu) = enqooqsfxk jiihsdtmdk (kvsmoywqor ) View more | ||||||
Not Applicable | - | zspkzmxbnt(qelywtmppc) = devlzjxxdm xxcibomwza (aqjxjkxmof ) | - | 02 Aug 2021 | |||
Non-Thymosin Alpha 1 | zspkzmxbnt(qelywtmppc) = hepcurawbf xxcibomwza (aqjxjkxmof ) | ||||||
Not Applicable | - | R-CHOP plus thymosin α1 | uzoqrsennr(yahvahijed) = ohiwipuisq qgccqfxpcr (jbtkrgydvf ) View more | Positive | 07 Jun 2017 | ||
R-CHOP | uzoqrsennr(yahvahijed) = djyzjkgnbi qgccqfxpcr (jbtkrgydvf ) View more | ||||||
Phase 3 | Hepatitis C, Chronic Adjuvant | 552 | Thymosin alpha-1 + Peginterferon alfa-2a/Ribavirin | avxexykesq(kyeaizhbte) = pmjdcgmkmh asysoegmyb (dqzezfysml ) | - | 01 Jan 2012 | |
Placebo + Peginterferon alfa-2a/Ribavirin | avxexykesq(kyeaizhbte) = gzxunrmeyg asysoegmyb (dqzezfysml ) | ||||||
Phase 2 | 488 | (Dacarbazin + Interferon Alpha + Thymosin-alpha-1 1.6 mg) | ibfrmwtzal = npbsafaojt sgkysgbvay (ipigqurxmm, lxcowuaqoy - qodsjxsdvr) View more | - | 02 Jun 2009 | ||
(Dacarbazin + Interferon Alpha + Thymosin-alpha-1 3.2 mg) | ibfrmwtzal = zrdfovpqww sgkysgbvay (ipigqurxmm, pqgbwoabnt - wsjnqbuxho) View more | ||||||
Not Applicable | 18 | (Group 1) | hbqziklrer(jwcedpmxjg) = gxwzonryur hdieegimfu (pjymofoxvo ) | - | 01 Jun 2005 | ||
(Group 2) | unqpeyiuuf(xsndwcmuwz) = astkqthelc epicemijhm (mixpgpvenw ) |