Last update 21 Nov 2024

Ezobresib

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
(S)-2-(3-(1,4-dimethyl-1H-1,2,3-triazol-5-yl)-5-(phenyl(tetrahydro-2H-pyran-4-yl)methyl)-5H-pyrido[3,2-b]indol-7-yl)propan-2-ol, 2-(3-(3,5-Dimethyltriazol-4-yl)-5-((S)-oxan-4-yl(phenyl)methyl)pyrido(3,2-b)indol-7-yl)propan-2-ol
+ [1]
Target
Mechanism
BET inhibitors(Bromodomain and extra terminal domain protein inhibitors)
Originator Organization
Inactive Organization-
Drug Highest PhasePhase 2
First Approval Date-
RegulationOrphan Drug (EU)
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Structure

Molecular FormulaC30H33N5O2
InChIKeyKGERZPVQIRYWRK-GDLZYMKVSA-N
CAS Registry1800340-40-2

External Link

KEGGWikiATCDrug Bank
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R&D Status

10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
Advanced cancerPhase 2
CA
19 Jun 2015
Advanced Malignant Solid NeoplasmPhase 2
ES
19 Jun 2015
Advanced Malignant Solid NeoplasmPhase 2
FR
19 Jun 2015
Advanced Malignant Solid NeoplasmPhase 2
CA
19 Jun 2015
Advanced Malignant Solid NeoplasmPhase 2
US
19 Jun 2015
Advanced Malignant Solid NeoplasmPhase 2
AU
19 Jun 2015
Advanced cancerPreclinical
FR
19 Jun 2015
Advanced cancerPreclinical
ES
19 Jun 2015
Advanced cancerPreclinical
AU
19 Jun 2015
Advanced cancerPreclinical
US
19 Jun 2015
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Phase 1/2
40
(roasgnvkqs) = nmviradqia kdieggascu (siovhhmkth )
-
10 Dec 2023
(roasgnvkqs) = ecepvxdvnv kdieggascu (siovhhmkth )
Phase 1/2
13
(ydaorypfhm) = eflichtxfg anorugzqtu (bcbbsvtvxj )
Positive
15 Nov 2022
(ydaorypfhm) = fjcyghrjxk anorugzqtu (bcbbsvtvxj )
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Approval

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Regulation

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