Last update 20 Mar 2025

Lunresertib

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
Target
Action
inhibitors
Mechanism
PKMYT1 inhibitors(protein kinase, membrane associated tyrosine/threonine 1 inhibitors)
Inactive Indication-
Originator Organization
Inactive Organization-
Drug Highest PhasePhase 2
First Approval Date-
RegulationFast Track (United States)
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Structure/Sequence

Molecular FormulaC18H20N4O2
InChIKeyARBRHWRTXPWZGN-UHFFFAOYSA-N
CAS Registry2719793-90-3

R&D Status

10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
Colorectal CancerPhase 2
Canada
24 May 2023
Colorectal CancerPhase 2
Canada
24 May 2023
Neoplasm MetastasisPhase 2
Canada
24 May 2023
Neoplasm MetastasisPhase 2
Canada
24 May 2023
Ovarian CancerPhase 2
Canada
24 May 2023
Ovarian CancerPhase 2
Canada
24 May 2023
Ovarian CarcinosarcomaPhase 2
Canada
24 May 2023
Ovarian CarcinosarcomaPhase 2
Canada
24 May 2023
Primary peritoneal carcinomaPhase 2
Canada
24 May 2023
Primary peritoneal carcinomaPhase 2
Canada
24 May 2023
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Phase 1
51
(Endometrial Cancer)
(bnpggdckyd) = iahczobmnw hhxdpagrtr (lscwnrlfsk )
Positive
12 Dec 2024
(Platinum-Resistant Ovarian Cancer)
(bnpggdckyd) = idlmhiivrk hhxdpagrtr (lscwnrlfsk )
Phase 1
38
Lunresertib + FOLFIRI
(gastrointestinal cancers)
(mgdljbzgwe) = Neutropenia and leukopenia ljowvoereh (oiwpmuljnm )
Positive
26 Jun 2024
Lunresertib + FOLFIRI
(CRC)
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Approval

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Regulation

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