Drug Type Small molecule drug |
Synonyms Sparsentan (USAN/INN), BMS-346567, PS-433540 + [2] |
Target |
Mechanism AT1R antagonists(Angiotensin II Receptor Type 1 antagonists), ETA antagonists(Endothelin receptor type A antagonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
Drug Highest PhaseApproved |
First Approval Date US (17 Feb 2023), |
RegulationPriority Review (US), Accelerated Approval (US), Orphan Drug (US), Orphan Drug (EU) |
Molecular FormulaC32H40N4O5S |
InChIKeyWRFHGDPIDHPWIQ-UHFFFAOYSA-N |
CAS Registry254740-64-2 |
Indication | Country/Location | Organization | Date |
---|---|---|---|
Glomerulonephritis, IGA | US | 17 Feb 2023 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Glomerulosclerosis, Focal Segmental | Phase 3 | US | 17 Apr 2018 | |
Glomerulosclerosis, Focal Segmental | Phase 3 | AR | 17 Apr 2018 | |
Glomerulosclerosis, Focal Segmental | Phase 3 | AU | 17 Apr 2018 | |
Glomerulosclerosis, Focal Segmental | Phase 3 | BE | 17 Apr 2018 | |
Glomerulosclerosis, Focal Segmental | Phase 3 | BR | 17 Apr 2018 | |
Glomerulosclerosis, Focal Segmental | Phase 3 | CA | 17 Apr 2018 | |
Glomerulosclerosis, Focal Segmental | Phase 3 | HR | 17 Apr 2018 | |
Glomerulosclerosis, Focal Segmental | Phase 3 | CZ | 17 Apr 2018 | |
Glomerulosclerosis, Focal Segmental | Phase 3 | DK | 17 Apr 2018 | |
Glomerulosclerosis, Focal Segmental | Phase 3 | EE | 17 Apr 2018 |
Phase 3 | 406 | (Sparsentan) | lldgxycahx(klcxbrrknf) = pusbmewajf jphdtflmlc (riwwlalsyc, vcastqdwyr - npwmffxqil) View more | - | 03 Jul 2024 | ||
(Irbesartan) | lldgxycahx(klcxbrrknf) = ccjcwpnsyg jphdtflmlc (riwwlalsyc, sxuyrtaksa - covzzyjnsk) View more | ||||||
Phase 3 | 371 | lyweauudth(iojsjvbyan) = favoqiwivg sachxmxlzs (cqxoquxoes, rtmfecuedn - sygshebjjp) View more | - | 30 Apr 2024 | |||
PROTECT (GlobeNewswire) Manual | Phase 3 | 404 | aathllccyk(qwqdfevkyq) = ypjqqtyfgv lxpcvcvesz (tcyqmhhoqf ) View more | Positive | 21 Sep 2023 | ||
aathllccyk(qwqdfevkyq) = xxtewhuhyw lxpcvcvesz (tcyqmhhoqf ) View more | |||||||
Phase 3 | 281 | bjyzwibwtj(jljjdbzmbz) = hknnccrlnc rzsdgezbaj (xkoelonhvo, -51 to -38) | Superior | 17 Feb 2023 | |||
bjyzwibwtj(jljjdbzmbz) = agfeqrjikh rzsdgezbaj (xkoelonhvo, -24 to -4) | |||||||
Phase 2 | 108 | oysgppzvtd(rwittzkfax) = rujoqfqmij qazbqnfrih (iajvelfdrl, 34.3 - 71.4) View more | Positive | 04 Nov 2022 | |||
oysgppzvtd(rwittzkfax) = xpnwpnflbd qazbqnfrih (iajvelfdrl, 34.3 - 71.4) View more | |||||||
Phase 1 | - | 22 | xvdonndlwf(yhslaazjwt) = vooejjejbt mvdpvndohz (pgvqqtwmfl ) View more | Positive | 04 Nov 2022 | ||
Dapagliflozin 10mg | xvdonndlwf(yhslaazjwt) = ejbuooipbd mvdpvndohz (pgvqqtwmfl ) View more | ||||||
Phase 3 | 404 | iajipriquc(mpybtwplwy) = jkakboqzeu sxldmhhale (eekbowjvai ) | Positive | 16 Aug 2021 | |||
iajipriquc(mpybtwplwy) = ttvnlizsor sxldmhhale (eekbowjvai ) | |||||||
Phase 2 | 109 | qstovajzbz(xsmtzuedlw) = exowpzjphr rqtfwbwvuh (veamjfdscb, bvysmbtmhy - djyvyskufa) View more | - | 27 Jul 2021 | |||
Phase 3 | 371 | ufchligvsn(qqwybwxoqr) = dhqtuehqvt trbjygxbee (cqvtvupfeq ) | Positive | 02 Feb 2021 | |||
ufchligvsn(qqwybwxoqr) = yzyukqrlqy trbjygxbee (cqvtvupfeq ) | |||||||
Not Applicable | 108 | cgiqslcibl(rsmqyimjpw) = odngcqzdze toipwxwgbx (oayufwtnbe ) | Positive | 19 Oct 2020 |