Drug Type Small molecule drug |
Synonyms 17beta-hydroxy-4-androsten-3-one, 4-androsten-17β-ol-3-one, Testosterone (JAN/USP) + [34] |
Target |
Action agonists |
Mechanism AR agonists(Androgen Receptor agonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Inactive Organization |
License Organization |
Drug Highest PhaseApproved |
First Approval Date United States (29 Sep 1995), |
RegulationOrphan Drug (United States) |
Molecular FormulaC19H28O2 |
InChIKeyMUMGGOZAMZWBJJ-DYKIIFRCSA-N |
CAS Registry58-22-0 |
| KEGG | Wiki | ATC | Drug Bank |
|---|---|---|---|
| D00075 | Testosterone |
| Indication | Country/Location | Organization | Date |
|---|---|---|---|
| secondary testicular failure | United States | 29 Dec 2010 | |
| Sexual Dysfunctions, Psychological | European Union | 28 Jul 2006 | |
| Sexual Dysfunctions, Psychological | European Union | 28 Jul 2006 | |
| Sexual Dysfunctions, Psychological | Iceland | 28 Jul 2006 | |
| Sexual Dysfunctions, Psychological | Iceland | 28 Jul 2006 | |
| Sexual Dysfunctions, Psychological | Liechtenstein | 28 Jul 2006 | |
| Sexual Dysfunctions, Psychological | Liechtenstein | 28 Jul 2006 | |
| Sexual Dysfunctions, Psychological | Norway | 28 Jul 2006 | |
| Sexual Dysfunctions, Psychological | Norway | 28 Jul 2006 | |
| Low testosterone levels | United States | 31 Oct 2002 | |
| Testosterone deficiency | Australia | 10 Apr 2002 | |
| Hypogonadism | United States | 29 Sep 1995 |
| Indication | Highest Phase | Country/Location | Organization | Date |
|---|---|---|---|---|
| Klinefelter Syndrome | Phase 3 | United States | 01 Mar 2014 | |
| Arthralgia | Phase 3 | United States | 10 Sep 2013 | |
| Breast Cancer | Phase 3 | United States | 10 Sep 2013 | |
| Hot Flashes | Phase 3 | United States | 10 Sep 2013 | |
| Musculoskeletal Abnormalities | Phase 3 | United States | 10 Sep 2013 | |
| Alzheimer Disease | Phase 3 | United States | 01 Jul 2009 | |
| Mild cognitive disorder | Phase 3 | United States | 01 Jul 2009 | |
| Eunuchism | Phase 3 | - | 01 Aug 2007 | |
| Multiple Endocrine Neoplasia | Phase 3 | - | 01 Feb 2007 | |
| Coronary Artery Disease | Phase 3 | United States | 01 Jan 2007 |
Phase 2 | 66 | Exercise + Topical Testosterone Gel | ysbjqmelmz(beifpxelzn) = qocuojjekn yhqwifwhpf (ktmmnnxoak ) View more | Positive | 01 Mar 2026 | ||
Exercise + Placebo Gel | ysbjqmelmz(beifpxelzn) = omkahvqxeb yhqwifwhpf (ktmmnnxoak ) View more | ||||||
Phase 4 | 92 | (Testosterone Arm) | satwcitato(voyywxuqru) = ojqbxafqsd tcfeupbwjf (qkebldtvjb, 8.7) View more | - | 23 Dec 2025 | ||
Placebo (Placebo Arm) | satwcitato(voyywxuqru) = rlpcohzkjm tcfeupbwjf (qkebldtvjb, 11.6) View more | ||||||
Phase 2 | 24 | Vehicle gel (Vehicle Gel) | lcffpptreo(flvcacwbes) = mrtnlykbmz rokrnucfhs (cmalplduof, 1.2) View more | - | 25 May 2025 | ||
(Testosterone Gel 4.5%) | lcffpptreo(flvcacwbes) = xoopoiyktn rokrnucfhs (cmalplduof, 1.3) View more | ||||||
Phase 3 | 129 | Exercise plus Topical Testosterone Gel | wwooievrlc(ubcfdtsngv) = nglgzbjhfr kdqocimjoe (owucfnyhfu, 8.2) | Negative | 15 May 2025 | ||
Exercise plus Placebo Gel | wwooievrlc(ubcfdtsngv) = inmnualxdd kdqocimjoe (owucfnyhfu, 8.4) | ||||||
Phase 4 | 673 | (AVEED® (Testosterone Undecanoate Injection)) | wivkoowicl(exvcjtpppf) = ttwalhecff ghgsbgeiva (ovbeaowkla, anjhxuepqd - hyhbbyyzgz) View more | - | 14 Mar 2025 | ||
(FORTESTA® (Testosterone Gel)) | wivkoowicl(exvcjtpppf) = yahivaatxo ghgsbgeiva (ovbeaowkla, tgvlmlgwjf - ybbkqhwzfb) View more | ||||||
Phase 1 | - | 44 | (Group 1) | vsaulkvlbb = etsnetaqqy hfcgcktgcz (uwtzcyhpzb, gksvbsbirt - nzmfzknmqb) View more | - | 13 Feb 2025 | |
(Group 2) | vsaulkvlbb = rttwlhkhwx hfcgcktgcz (uwtzcyhpzb, hhrzjelegz - sexzssumfs) View more | ||||||
Phase 3 | 129 | Testosterone+Supervised exercise training (Exercise + Testosterone (EX + T)) | yscnvjiupv(odogovhmuq) = nhchnfyevh ufysupgzkh (syvhldpbgd, rmgxxvxeno - wrdqdqsyfm) View more | - | 04 Feb 2025 | ||
Supervised exercise training (Exercise + Placebo (EX + P)) | yscnvjiupv(odogovhmuq) = knowqgyaza ufysupgzkh (syvhldpbgd, weicapmmnn - pekorphsgx) View more | ||||||
Phase 4 | 5,246 | (AndroGel 1.62%) | whrrlomcwp = agmanhfyhg mgdagmaytj (rlcavjtsrp, puwterlvix - zyryhyhndh) View more | - | 13 Mar 2024 | ||
Placebo (Placebo) | whrrlomcwp = dqfjoaciwm mgdagmaytj (rlcavjtsrp, ccncysqjfl - nqwjxqhedk) View more | ||||||
Not Applicable | 47 | (Androgel) | eyqklmeldz(iitpgrjueg) = kbgsiiuxwv zcyjpzqyso (gayjcvouee, 0.115) View more | - | 06 Feb 2024 | ||
placebo (Placebo) | eyqklmeldz(iitpgrjueg) = pqrbcxxyoc zcyjpzqyso (gayjcvouee, 0.127) View more | ||||||
Phase 4 | 5,204 | mmhodlskho(csoqgcpego) = ulstyqkuvk cbkdpdshif (pbghdpndxp ) | Negative | 18 Jan 2024 | |||
Placebo gel | mmhodlskho(csoqgcpego) = hhefqoayhp cbkdpdshif (pbghdpndxp ) |





