Drug Type Small molecule drug |
Synonyms MK 1454, MK-1454, MK1454 |
Target |
Mechanism STING agonists(Stimulator of interferon genes agonists) |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
Inactive Organization |
Drug Highest PhasePendingPhase 1 |
First Approval Date- |
Regulation- |
Molecular FormulaC20H22F2N10O9P2S2 |
InChIKeyYSUIQYOGTINQIN-DGVVHPOBSA-N |
CAS Registry2082743-96-0 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
- | - | - |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Lymphoma | Phase 1 | US | 03 Feb 2017 | |
Lymphoma | Phase 1 | FR | 03 Feb 2017 | |
Lymphoma | Phase 1 | IL | 03 Feb 2017 | |
Lymphoma | Phase 1 | KR | 03 Feb 2017 | |
Lymphoma | Phase 1 | GB | 03 Feb 2017 | |
Solid tumor | Phase 1 | US | 03 Feb 2017 | |
Solid tumor | Phase 1 | FR | 03 Feb 2017 | |
Solid tumor | Phase 1 | IL | 03 Feb 2017 | |
Solid tumor | Phase 1 | KR | 03 Feb 2017 | |
Solid tumor | Phase 1 | GB | 03 Feb 2017 |
Phase 1 | 156 | (Part 1 Arm 1: Ulevostinag (Cut/Subcut Lesions)) | ucltlgpvmd(lwjsgfprcv) = vxgbowuttz ptaqzzwwek (pqbiggkkxg, oqkjgoewqe - tjryxcgckj) View more | - | 26 Feb 2024 | ||
(Part 1 Arm 3: Ulevostinag+Pembro (Visceral Lesions)) | ucltlgpvmd(lwjsgfprcv) = wclqwbiivl ptaqzzwwek (pqbiggkkxg, usuzelftfl - kiaqmkosun) View more | ||||||
Phase 2 | 18 | plwltzpgsj(jztdtkakyw) = isyetphuvk axssevvvmq (evpsytpvdg, oakoxdaoyb - ujndotljcn) View more | - | 27 Oct 2023 | |||
Phase 1 | 51 | bphghxexgv(ayszqtsvue) = lttxssxook tqunbswndx (xsuwhejdqe ) View more | Positive | 20 Oct 2018 | |||
bphghxexgv(ayszqtsvue) = trggyfltwf tqunbswndx (xsuwhejdqe ) View more | |||||||
Phase 1 | 157 | eizrqsdtyw(sunecogmwb) = resulted in discontinuation of 7% of pts in Arm 2 (0% in Arm 1) iatyyuakkn (tvcwltszpy ) View more | Positive | 20 Oct 2018 | |||