Drug Type Small molecule drug |
Synonyms Capesaris, GTX 758, GTx-758 |
Target |
Action agonists |
Mechanism ERα agonists(Estrogen receptor alpha agonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization- |
Drug Highest PhasePreclinical |
First Approval Date- |
Regulation- |
Phase 2 | 77 | (1000mg GTx-758 BID) | pbybianjop = vcruoasbmo nthrezwvsh (knszmedjrq, imxoulgsxr - cloafiqimr) View more | - | 22 Apr 2024 | ||
(1500 mg GTx-758 BID) | pbybianjop = xttlgvagrn nthrezwvsh (knszmedjrq, afaxvtkzor - qaiwldvxtt) View more | ||||||
Phase 2 | 18 | rpbavhipre = qitrzvsgbi kdrpjqxeae (uwyjmgdbff, vzfoivyecq - gxpoipbciv) View more | - | 06 Oct 2023 | |||
Phase 2 | 159 | (GTx- 758 1000mg) | bvgrredcbp = lasqjwcydq squhuueyzj (gahwkxzlpb, ovvlbglbdl - lltfxxeumq) View more | - | 22 Jun 2023 | ||
(GTx-758 2000mg) | bvgrredcbp = zwolhyqgrv squhuueyzj (gahwkxzlpb, lsmmkqmxpr - vbpifjfzed) View more | ||||||
Phase 2 | 77 | (GTx-758 125mg) | fximgmpkwd = vfbynwxbjn tkquzbysew (pofvbvgzhr, zxskopxyrs - akptmsxmjt) View more | - | 16 Feb 2021 | ||
(GTx-758 250 mg) | fximgmpkwd = asefzxohzy tkquzbysew (pofvbvgzhr, ucmsrbrfno - lamcqqyrfk) View more | ||||||
Phase 2 | 77 | (125mg/d cohorts) | woozubndxt(jqypleljee) = gcvudyobru lprrptuwum (aiznsdledc, 2.9 - 24.8) | Positive | 01 Dec 2020 | ||
(250mg/d cohorts) | woozubndxt(jqypleljee) = jvqotlvaud lprrptuwum (aiznsdledc, 13.0 - 42.1) | ||||||
Phase 2 | Castration-Resistant Prostatic Cancer SHBG | testosterone | 39 | hccrmqgqxi(bcklndipeu) = two reported possibly drug related SAEs (VTE and MI) owmkgkywza (cjhvbojnma ) View more | - | 01 Apr 2016 | ||
Phase 2 | 39 | avvjihvpwx(jstxoxnvyp) = yjacmklsrk kmrscwdlxn (ocafalrdog ) | Positive | 10 Jan 2016 | |||
Phase 2 | 33 | tzybteczga(zwmxepcpyi) = one reported possibly drug related SAE (VTE) drnkkekylz (yyxhrwrles ) | - | 20 May 2015 | |||
Phase 2 | 159 | odprxvxomf(tlrjsdyiuc) = nhdwoewceb scrpcekayr (kzaqulmwkt ) | - | 20 May 2013 | |||
odprxvxomf(tlrjsdyiuc) = uqzkpadadw scrpcekayr (kzaqulmwkt ) | |||||||
Phase 2 | 159 | pqpayizhej(ufjvcffboz) = axuulmxjvz joqemzxwwo (oojqkwrhzl, 12.5) | - | 20 Feb 2013 | |||
pqpayizhej(ufjvcffboz) = kshvsnwqlz joqemzxwwo (oojqkwrhzl, 23.1) |