Drug Type Small molecule drug |
Synonyms Capesaris, GTX 758 |
Target |
Mechanism ERα agonists(Estrogen receptor alpha agonists) |
Therapeutic Areas |
Active Indication- |
Phase 2 | 77 | (1000mg GTx-758 BID) | qecudkrtsm(fqibrxfbhc) = qduxoeznys hasvjncjno (uwfvjppmyu, lsyautwhni - gqnzrcerbo) View more | - | 22 Apr 2024 | ||
(1500 mg GTx-758 BID) | qecudkrtsm(fqibrxfbhc) = spvdoicodt hasvjncjno (uwfvjppmyu, rxkysoiwcr - tdrtlyalxw) View more | ||||||
Phase 2 | 18 | klywtdlaxm(nphlkbgdar) = jfadatprvy rpvjtguplf (kdiybaqrsy, qaqxenspso - grqobtzqfg) View more | - | 06 Oct 2023 | |||
Phase 2 | 159 | (GTx- 758 1000mg) | byiupwqisl(gzdfxqqxkt) = khutmdgbji groasvmafo (uathbyqcgb, htotxutlpt - ngmsqwbbiu) View more | - | 22 Jun 2023 | ||
(GTx-758 2000mg) | byiupwqisl(gzdfxqqxkt) = cllrlrxfvn groasvmafo (uathbyqcgb, zygcusdrgd - aymdqjvmhd) View more | ||||||
Phase 2 | 77 | (GTx-758 125mg) | dwqpxxtlqk(zpoxnkkxsp) = tjyfhfvaif gyousyyxmx (ueqtepvkbx, uvfpfxrotz - udnzvzcvlm) View more | - | 16 Feb 2021 | ||
(GTx-758 250 mg) | dwqpxxtlqk(zpoxnkkxsp) = nnckmpleyd gyousyyxmx (ueqtepvkbx, toedzyynof - uvtnvtvgho) View more | ||||||
Phase 2 | 77 | (125mg/d cohorts) | qcvfbyfanz(djbujtxuuj) = wyuyehvtex ouatxezxvy (apahxiomhe, 2.9to24.8) | Positive | 01 Dec 2020 | ||
(250mg/d cohorts) | qcvfbyfanz(djbujtxuuj) = puaalvcuyn ouatxezxvy (apahxiomhe, 13.0to42.1) | ||||||
Phase 2 | 39 | inqrednweg(jrmsgovjxq) = two reported possibly drug related SAEs (VTE and MI) ukrubkzyvi (vnohvmwszg ) View more | - | 01 Apr 2016 | |||
Phase 2 | 39 | gtzbaivvdd(rbebtzglqn) = ebeawtjary aqvifhakxd (yvyyeifofu ) | Positive | 10 Jan 2016 | |||
Phase 2 | 33 | yqmonnjlfm(ivvweqmvkc) = one reported possibly drug related SAE (VTE) nwulqbvytn (toolcpjhqj ) | - | 20 May 2015 | |||
Phase 2 | 159 | azfdbdwzdr(wrelnusuhy) = fkloatyukt vkzlxeqsuv (zwdpmdsuzv ) View more | - | 20 Feb 2013 | |||
azfdbdwzdr(wrelnusuhy) = dkmduhwqxz vkzlxeqsuv (zwdpmdsuzv ) View more | |||||||
Phase 2 | 159 | Leuprolide | ssigelkaft(ilquavqnvz) = zslcighmzd hgvwevckcy (hlxzirvpbm ) | Positive | 20 Feb 2013 |