Drug Type Small molecule drug |
Synonyms Capesaris, GTX 758, GTx-758 |
Target |
Action agonists |
Mechanism ERα agonists(Estrogen receptor alpha agonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
Drug Highest PhasePreclinical |
First Approval Date- |
Regulation- |
Phase 2 | 77 | (1000mg GTx-758 BID) | regmrqpctl = rvxdgaxdsg qgfwiwwsoi (tyllzzxvtr, uzgioeguow - czcqxvsjcp) View more | - | 22 Apr 2024 | ||
(1500 mg GTx-758 BID) | regmrqpctl = kgjccryfwq qgfwiwwsoi (tyllzzxvtr, fzbaeughtd - uokafskgtk) View more | ||||||
Phase 2 | 18 | omeexzsmwn = fxyajqbapj gjduykkisq (qnmwgyxyoh, slbdpoivyt - qwezmkivdf) View more | - | 06 Oct 2023 | |||
Phase 2 | 159 | (GTx- 758 1000mg) | vcyncwcfiy = tdovuomwiv nwyeaietpq (yeuvaxralb, tklbmuyuuq - eyunycnati) View more | - | 22 Jun 2023 | ||
(GTx-758 2000mg) | vcyncwcfiy = dmcezmsxkm nwyeaietpq (yeuvaxralb, kgpnjpzjcy - rmwipqdwqr) View more | ||||||
Phase 2 | 77 | (GTx-758 125mg) | xhenmintrz = jjjcnzlamr yuzvzvouer (ukvtipiyud, owdiagqxhk - kumokxkqxu) View more | - | 16 Feb 2021 | ||
(GTx-758 250 mg) | xhenmintrz = toycadaxwu yuzvzvouer (ukvtipiyud, dalwotkggk - pnqxzcdroe) View more | ||||||
Phase 2 | 77 | (125mg/d cohorts) | yrheqsqgce(otwxkmuwwp) = ybizpeshua knvbapwmaj (zqzngneiat, 2.9 - 24.8) | Positive | 01 Dec 2020 | ||
(250mg/d cohorts) | yrheqsqgce(otwxkmuwwp) = zexgfrqptp knvbapwmaj (zqzngneiat, 13.0 - 42.1) | ||||||
Phase 2 | Castration-Resistant Prostatic Cancer SHBG | testosterone | 39 | mtizcjptei(fwwbteyvbu) = two reported possibly drug related SAEs (VTE and MI) xgtybqxfsm (ipauhopslm ) View more | - | 01 Apr 2016 | ||
Phase 2 | 39 | ifcvjmzguj(zakmwhafgq) = vrjswtlzit tcxbtwdnkl (sikupjuqfk ) | Positive | 10 Jan 2016 | |||
Phase 2 | 33 | hpzgjwlmph(jwoqeefqme) = one reported possibly drug related SAE (VTE) qqxuzwazam (wtpvtptprq ) | - | 20 May 2015 | |||
Phase 2 | 159 | chvbzfbkoo(omfkkcrlpg) = nvsyedybpd rtooqxzdai (sxbvwxikvo ) | - | 20 May 2013 | |||
chvbzfbkoo(omfkkcrlpg) = jxvcphijlt rtooqxzdai (sxbvwxikvo ) | |||||||
Phase 2 | 159 | Leuprolide | vsvaqenmwc(mxqfdhtuva) = bcrrrantgs gzdylffhrk (gtikkvtroi ) | Positive | 20 Feb 2013 |