[Translation] A Phase I Dose-Escalation Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Preliminary Efficacy of Oral YY2201 Tablets in Patients with Advanced Solid Tumors
主要目的:评估口服 YY2201在晚期实体瘤患者中的安全性和耐受性;评估口服 YY2201在晚期实体瘤患者中的最大耐受剂量(MTD)和/或Ⅱ期推荐剂量(RP2D);
次要目的:评估 YY2201在晚期实体瘤患者中的药代动力学(PK)特征;初步评估口服 YY2201在晚期实体瘤患者中的抗肿瘤疗效。
[Translation] Primary objectives: To evaluate the safety and tolerability of oral YY2201 in patients with advanced solid tumors; To evaluate the maximum tolerated dose (MTD) and/or phase II recommended dose (RP2D) of oral YY2201 in patients with advanced solid tumors;
Secondary objectives: To evaluate the pharmacokinetic (PK) characteristics of YY2201 in patients with advanced solid tumors; To preliminarily evaluate the anti-tumor efficacy of oral YY2201 in patients with advanced solid tumors.