Author: Nijmeijer, Saskia ; Istyastono, Enade P. ; de Graaf, Chris ; de Esch, Iwan J. P. ; Smits, Rogier A. ; Vischer, Henry F. ; Kooistra, Albert J. ; Leurs, Rob ; Roumen, Luc ; Kuijer, Martien
Structure-based virtual screening using H1R- and β2R-based histamine H4R homology models identified 9 fragments with an affinity ranging from 0.14 to 6.3 μm for H4R.