Last update 31 May 2024

Uzansertib

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
INCB-053914, INCB-53914
Mechanism
PIM1 inhibitors(Proto-oncogene serine/threonine-protein kinase Pim-1 inhibitors), PIM2 inhibitors(Serine/threonine-protein kinase pim-2 inhibitors), PIM3 inhibitors(Serine/threonine-protein kinase pim-3 inhibitors)
Active Indication-
Originator Organization
Active Organization-
Drug Highest PhaseDiscontinuedPhase 1/2
First Approval Date-
Regulation-

Structure

Molecular FormulaC26H26F3N5O3
InChIKeyPTORCEYGCGXHDH-OVMXCRKPSA-N
CAS Registry1620012-39-6

R&D Status

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IndicationHighest PhaseCountry/LocationOrganizationDate
Solid tumorPhase 2
US
29 Dec 2015
Plasma cell myeloma refractoryPhase 1-01 Jul 2021
Relapse multiple myelomaPhase 1-01 Jul 2021
Diffuse large B-cell lymphoma recurrentPhase 1
US
03 Dec 2018
Diffuse large B-cell lymphoma refractoryPhase 1
US
03 Dec 2018
Acute Myeloid LeukemiaPreclinical
US
-
Multiple MyelomaPreclinical
US
-
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Phase 1/2
39
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Positive
07 Dec 2017
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Deal

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Clinical Trial

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Approval

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Regulation

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