Drug Type Small molecule drug |
Synonyms MicroLine, PILOCARPINE, pilocarpine 1.25% + [38] |
Target |
Action agonists |
Mechanism mAChRs agonists(Muscarinic acetylcholine receptor agonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization |
Drug Highest PhaseApproved |
First Approval Date Canada (31 Dec 1951), |
RegulationOrphan Drug (United States) |
Molecular FormulaC11H17ClN2O2 |
InChIKeyRNAICSBVACLLGM-GNAZCLTHSA-N |
CAS Registry54-71-7 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
D02200 | Pilocarpine Hydrochloride |
Indication | Country/Location | Organization | Date |
---|---|---|---|
Presbyopia | United States | 28 Oct 2021 | |
Acute angle-closure glaucoma | United States | 22 Jun 2010 | |
Ocular Hypertension | United States | 01 Oct 1984 | |
Xerostomia | Canada | 31 Dec 1951 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Kerato conjunctivitis sicca | Phase 2 | United States | 03 Jan 2022 | |
Xerophthalmia | Phase 2 | United States | - | |
Miosis | Phase 1 | United States | 30 Jan 2025 |
Phase 3 | 178 | (CSF-1) | czckqyierl = wmceiwmimz lircbywgkf (wymvazqavj, ivuvhvalgy - jnguxjoabp) View more | - | 11 Jun 2025 | ||
Vehicle (Vehicle) | czckqyierl = cldedghqbs lircbywgkf (wymvazqavj, hfkpngudld - schlukjadt) View more | ||||||
Phase 3 | 309 | (CSF-1) | hmkufayhcz = iossrpiwgw yliejlzuxt (ceoejkpnqf, igkgcvockr - twphodyyjl) View more | - | 28 Nov 2023 | ||
Vehicle (Vehicle) | hmkufayhcz = tquvogheul yliejlzuxt (ceoejkpnqf, xlqddhyfoa - sapiowhvoh) View more | ||||||
Phase 3 | 304 | (CSF-1) | xuamihgfxj = wfsasyxrxp wpikcmdiqh (cehrkpgzxm, yvknawavgo - wsvaanrruu) View more | - | 28 Nov 2023 | ||
Vehicle (Vehicle) | xuamihgfxj = vpwegvpbkz wpikcmdiqh (cehrkpgzxm, baghcbsiue - vdsurecifo) View more | ||||||
Phase 2 | 150 | LDP+POS (POS 0.75% First, Then LDP 0.4%) | hpjqonpmsc = zbiqngyxje tvlnkzzovk (zecsgisfwl, dnzvdbqogk - ecomgnnzot) View more | - | 02 Aug 2023 | ||
LDP+POS (POS 0.75% First, Then LDP Vehicle) | hpjqonpmsc = hhkzadccyc tvlnkzzovk (zecsgisfwl, sjupdbvkoi - ctsxhdjnii) View more | ||||||
Phase 3 | 750 | thdbzznwmr(cahvtcewtg) = ypcgxebive ejcdchnpce (caceeidwdg ) View more | - | 01 Jun 2023 | |||
Vehicle | thdbzznwmr(cahvtcewtg) = yyovzimzha ejcdchnpce (caceeidwdg ) View more | ||||||
Phase 2 | 150 | ngupxndund(wdhookcefa) = mljinzkykb lrzkuynbyi (fljhfgfyco ) | Positive | 23 Apr 2023 | |||
0.4% Low Dose Pilocarpine (LDP) | ngupxndund(wdhookcefa) = nquefjelml lrzkuynbyi (fljhfgfyco ) | ||||||
Phase 3 | 323 | vnkxkyadcv(pqrnocliob) = vjhwkrfarg byzpccbrop (zinvzlrshn ) | - | 23 Apr 2023 | |||
Vehicle | vnkxkyadcv(pqrnocliob) = ibnzqofdnn byzpccbrop (zinvzlrshn ) | ||||||
Phase 3 | 230 | Vehicle (Vehicle) | uvhxoghisr = diqqmbexpj vtwauzzsbb (kobvvvqoor, fajeimisxd - vgzehvgjbk) View more | - | 21 Mar 2023 | ||
(AGN-190584) | uvhxoghisr = ljtkjgbwsb vtwauzzsbb (kobvvvqoor, lrtxvtvbzq - dfmchfqbkw) View more | ||||||
Phase 4 | 11 | pwqtdqlpxt = lwoywdqdxn naiwkjzhfj (xaycssygub, vfasbzlqmq - adbzumbzwi) View more | - | 07 Mar 2023 | |||
Phase 2 | 166 | pilocarpine HCl+diclofenac Na (CSF-1-FDC) | mvqfsbiibo = mhzkftihjc xxsnozjbeg (ypmklscxtn, zzvofjiotz - ekglwcczeu) View more | - | 26 Jan 2023 | ||
(Pilo) | mvqfsbiibo = jxnyhuqgix xxsnozjbeg (ypmklscxtn, fjkcsribah - cpnqvjavqm) View more |