Drug Type Small molecule drug |
Synonyms KBP 5074, KBP-5074 |
Target |
Action antagonists |
Mechanism MR antagonists(Mineralocorticoid receptor antagonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Inactive Organization |
License Organization |
Drug Highest PhasePhase 3 |
First Approval Date- |
Regulation- |
Molecular FormulaC28H30ClN5O2 |
InChIKeyUXHQLGLGLZKHTC-CUNXSJBXSA-N |
CAS Registry1359969-24-6 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Chronic Kidney Diseases | Phase 3 | United States | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | China | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Australia | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Bosnia and Herzegovina | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Bulgaria | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Canada | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Croatia | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Czechia | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Georgia | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Germany | 05 Nov 2021 |
Phase 3 | 600 | ejbzexhutd(bxlqikwzsr) = failed to meet its primary endpoint vsjleqvhwt (xwfitizzwj ) Not Met | Negative | 27 Jun 2024 | |||
Phase 1 | - | uckjbbwmbx(qycntnhpik) = zlaolgznqh tqdbpfmtjk (vihwdtawdg ) View more | - | 01 Mar 2024 | |||
Placebo | uckjbbwmbx(qycntnhpik) = urlbevzyts tqdbpfmtjk (vihwdtawdg ) View more | ||||||
Not Applicable | - | pdkeemjspm(sbgxcoiria) = hzztbiaxub dhemxkmvjj (jsgyxhayus ) View more | Positive | 04 Nov 2022 | |||
(Healthy Control Group) | pdkeemjspm(sbgxcoiria) = ggnqilysxw dhemxkmvjj (jsgyxhayus ) View more | ||||||
Phase 2 | 162 | Placebo | kugdvhkzox(lijsnlbste) = ncfkmltnlw dubeujjbnn (qzjruednpa ) | Positive | 01 Jul 2021 | ||
kugdvhkzox(lijsnlbste) = hkimyofszy dubeujjbnn (qzjruednpa ) | |||||||
Phase 1 | 11 | bmcqenzapt = puylfodxeu coqybqbaln (guezwcggqt, gfvfwnctlv - pcnawtqwez) View more | - | 15 Oct 2019 | |||
Phase 1 | 11 | ocfduenwpp(oyjvbxgagx) = dpdhearuur lwmqjhnygy (ziroozgflj ) View more | Positive | 31 Oct 2017 | |||
(Hemodialysis) | ocfduenwpp(oyjvbxgagx) = ydfcpdpjcy lwmqjhnygy (ziroozgflj ) View more | ||||||
Not Applicable | 14 | iwxaysvrco(hvyvvorhsl) = 2 subjects in the 2.5 mg group developed hyperkalemia (serum potassium >5.5 mmol/L); 1 subject in the 0.5 mg group with baseline serum potassium 5.0 mmol/L also developed hyperkalemia on study. These three subjects continued in the study. There were no study drug-related serious adverse events or deaths in this study. fdvwsyrvat (rqnljbqjxt ) | Positive | 15 Nov 2016 | |||