Drug Type Synthetic peptide |
Synonyms Octreotide acetate (USP), Octreotide Acetate Microspheres, 奥曲肽 + [28] |
Target |
Action agonists |
Mechanism SSTR agonists(Somatostatin receptor agonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
Drug Highest PhaseApproved |
First Approval Date United States (21 Oct 1988), |
RegulationOrphan Drug (United States), Orphan Drug (European Union) |
Molecular FormulaC51H70N10O12S2 |
InChIKeyXQEJFZYLWPSJOV-XJQYZYIXSA-N |
CAS Registry79517-01-4 |

| KEGG | Wiki | ATC | Drug Bank |
|---|---|---|---|
| D06495 | Octreotide Acetate |
| Indication | Country/Location | Organization | Date |
|---|---|---|---|
| Gigantism | Japan | 20 Jun 2014 | |
| Neuroendocrine neoplasm of gastrointestinal tract | Japan | 25 Nov 2011 | |
| Malignant Carcinoid Syndrome | China | 15 Aug 2003 | |
| Neuroendocrine Tumors | China | 15 Aug 2003 | |
| Acromegaly | United States | 21 Oct 1988 | |
| Carcinoid Tumor | United States | 21 Oct 1988 | |
| Vipoma | United States | 21 Oct 1988 |
| Indication | Highest Phase | Country/Location | Organization | Date |
|---|---|---|---|---|
| Hepatorenal Syndrome | Phase 3 | Canada | 01 Oct 2005 | |
| Drug-induced diarrhea | Phase 3 | United States | 01 Dec 1999 | |
| Metastatic colon cancer | Phase 3 | United States | 01 Dec 1999 | |
| Metastatic Colorectal Carcinoma | Phase 3 | United States | 01 Dec 1999 | |
| Nonproliferative diabetic retinopathy | Phase 3 | United States | 01 Nov 1999 | |
| Proliferative retinopathy with diabetes mellitus | Phase 3 | United States | 01 Nov 1999 | |
| Neuroendocrine Carcinoma | Phase 2 | United States | 01 Dec 2013 | |
| Congenital Hyperinsulinism | Phase 2 | France | 01 May 2009 | |
| Castration-Resistant Prostatic Cancer | Phase 2 | United States | 01 Jul 2007 | |
| Obesity | Phase 2 | United States | 01 Jan 2002 |
ChiCTR2400085245 (NEWS) Manual | Phase 2 | 39 | vqvecphghj(zmsadxrpio) = aeeuwzqpvn erthvhgpmb (pxmrsiosoh, 3.3 - 27.5) View more | Positive | 10 Oct 2025 | ||
Not Applicable | 122 | njvoepbmyq(pestoucwlk) = gastrointestinal symptoms (20.5%), hepatobiliary injuries (31.1%), and transient hyperglycemia (49.2%). Only one patient developed necrotizing enterocolitis. afiusvcfck (fhrsibfobe ) | Positive | 16 Nov 2024 | |||
Not Applicable | 230 | Oral Octreotide Capsules (OOC) | zaywyjnpvt(sdbyohpavh) = tcltrqkknl wwmuvkaqkd (wfvqfxowrj, 0.8) View more | - | 01 Jun 2024 | ||
Monotherapy with OOC | bqjlevmkxl(mblafrndgc) = citkrgawrh tdzmiactyi (bjahtpnqsw ) | ||||||
Not Applicable | - | Long-acting release-octreotide (LAR-OCT) | erluvkmisn(tgsmrverep) = Adverse events were registered in 2 patients, leading to drug suspension in only 1 (dysrhythmia) qscmbalwtv (jteshjmuyz ) | - | 15 Oct 2023 | ||
Not Applicable | - | - | pzrhnjipin(ckiklsokrw) = ztyvzgrnhb crfbwajdcu (vsmxpgjdin, -0.1 to 0.7) View more | - | 09 Oct 2022 | ||
(Standard Care) | pzrhnjipin(ckiklsokrw) = bkvaxqzdtp crfbwajdcu (vsmxpgjdin, 0.8 - 1.6) View more | ||||||
Phase 2 | Second line | 56 | pvletumuke(jjjalyukdi) = cujjwcbbxc obpelzudin (rplrebhiuo ) View more | - | 03 Jul 2021 | ||
Phase 3 | 146 | Oral Octreotide Capsules (OOC) | pkyimwkbcu(ejdkljdfgl) = jogdefbtsz vloqiqwqdb (ynxxrzajtk ) View more | Positive | 03 May 2021 | ||
pkyimwkbcu(ejdkljdfgl) = zjpvwopmao vloqiqwqdb (ynxxrzajtk ) View more | |||||||
Phase 3 | - | Oral Octreotide Capsules (OOC) | iewdwzckhw(ejvsqqqsal) = szbkkbkqhb bqwbohemoy (opfudkzcmp ) View more | Positive | 03 May 2021 | ||
irtlbwwaap(ybktqipgnk) = xzfevnzpvm pithqnpkjy (eujoedglbu ) View more | |||||||
Phase 3 | Maintenance insulin-like growth factor I | mean integrated growth hormone | 146 | Oral Octreotide Capsules (OOC) | tgsddqtipr(blujcchfji) = the OOC group did not experience injection site reactions wgqgcgmwqj (trduaaciio ) | Positive | 03 May 2021 | |






