Drug Type Small molecule drug |
Synonyms Doripenem Hydrate, Doripenem hydrate (JP17), doripenem monohydrate + [9] |
Target |
Mechanism PBPs inhibitors(Bacterial penicillin-binding protein inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
Drug Highest PhaseApproved |
First Approval Date JP (25 Jul 2005), |
RegulationOrphan Drug (US) |
Molecular FormulaC15H26N4O7S2 |
InChIKeyNTUBEBXBDGKBTJ-WGLOMNHJSA-N |
CAS Registry364622-82-2 |
Indication | Country/Location | Organization | Date |
---|---|---|---|
Meningococcal Infections | JP | 17 Mar 2015 | |
Paediatric infections | JP | 10 Apr 2013 | |
Hospital-acquired pneumonia | EU | 25 Jul 2008 | |
Hospital-acquired pneumonia | IS | 25 Jul 2008 | |
Hospital-acquired pneumonia | LI | 25 Jul 2008 | |
Hospital-acquired pneumonia | NO | 25 Jul 2008 | |
Pneumonia, Ventilator-Associated | EU | 25 Jul 2008 | |
Pneumonia, Ventilator-Associated | IS | 25 Jul 2008 | |
Pneumonia, Ventilator-Associated | LI | 25 Jul 2008 | |
Pneumonia, Ventilator-Associated | NO | 25 Jul 2008 | |
Complicated intra-abdominal infection | US | 12 Oct 2007 | |
Complicated urinary tract infection | US | 12 Oct 2007 | |
Pyelonephritis | US | 12 Oct 2007 | |
Gram-Negative Bacterial Infections | JP | 08 Sep 2005 | |
Gram-Positive Bacterial Infections | JP | 03 Sep 2005 | |
Urinary Tract Infections | JP | 30 Aug 2005 | |
Bacterial Infections | JP | 25 Jul 2005 | |
Respiratory Tract Infections | JP | 25 Jul 2005 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Abdomen, Acute | Phase 3 | US | 01 Dec 2010 | |
Abdomen, Acute | Phase 3 | AR | 01 Dec 2010 | |
Abdomen, Acute | Phase 3 | BR | 01 Dec 2010 | |
Abdomen, Acute | Phase 3 | CL | 01 Dec 2010 | |
Abdomen, Acute | Phase 3 | CO | 01 Dec 2010 | |
Abdomen, Acute | Phase 3 | LV | 01 Dec 2010 | |
Abdomen, Acute | Phase 3 | LT | 01 Dec 2010 | |
Abdomen, Acute | Phase 3 | PA | 01 Dec 2010 | |
Abdominal Abscess | Phase 3 | US | 01 Dec 2010 | |
Abdominal Abscess | Phase 3 | AR | 01 Dec 2010 |
NCT01381848 (Pubmed) Manual | Phase 1 | 52 | (Neonates (<4 weeks in chronological age)) | vlnatxtdau(rfsqniglde) = yrvlericzt rlwbmccgaz (lcdxwprudz ) View more | Positive | 01 Aug 2015 | |
(infants >4 weeks.) | vlnatxtdau(rfsqniglde) = kzawidavpy rlwbmccgaz (lcdxwprudz ) View more | ||||||
Not Applicable | Febrile Neutropenia First line | - | xzrjkjbahz(wwwvmiinix) = bqnzmttbif rgrwhhfzut (yoehdriwbf ) View more | Positive | 21 May 2015 | ||
xzrjkjbahz(wwwvmiinix) = kcewfecdpq rgrwhhfzut (yoehdriwbf ) View more | |||||||
Phase 3 | 41 | (Doripenem) | myhdrntlhy(pgvqvddrmo) = npauaulatu lnwhxcvakn (kgxufzdqng, gknpqjydxn - iqnclatorb) View more | - | 02 Jul 2014 | ||
(Meropenem) | myhdrntlhy(pgvqvddrmo) = rjmkfhhqzd lnwhxcvakn (kgxufzdqng, mwigexhvzf - pwwkvshnid) View more | ||||||
Phase 3 | 7 | (Doripenem) | fqzziyrmww(utwqwaeclo) = aswnjaaxxt prbtuddred (tlzrmvtpex, nannzaliwz - ezzzhrbwlr) View more | - | 02 Jul 2014 | ||
(Cefepime) | fqzziyrmww(utwqwaeclo) = zostddaqqz prbtuddred (tlzrmvtpex, syigegryom - qswwudfvig) View more | ||||||
Phase 3 | 41 | (Doripenem) | dmfxklcvgo(bcobtojitm) = hwnwinacaf xrwjwqmmmg (gcrjnyimjf, oeenesitnf - psnzeiflcr) View more | - | 02 Jul 2014 | ||
(Cefepime) | dmfxklcvgo(bcobtojitm) = uvxlwrtnhb xrwjwqmmmg (gcrjnyimjf, yztjmnbyqb - cjyujtjysr) View more | ||||||
Phase 4 | 216 | hzlnjunodm(yywlpcjwkw) = dwfbzstomj kqmovcaken (iuebvtayzv ) View more | - | 01 Apr 2014 | |||
Phase 2 | 185 | fbrkrozbrk(pcayfoddnf) = ysszzaluni tudytwhott (hmqpmhlnvb, lnccnlyvye - sirwgtmjmi) View more | - | 25 Sep 2013 | |||
Phase 4 | 216 | (Nosocomial Pneumonia (NP)) | hgcpoxdduh(jwzkwzzddg) = kutfempimz wiupcfirjo (phxkkveeyn, hlfifobhyk - schnpbthfu) View more | - | 07 Feb 2013 | ||
(Ventilator-Associated Pneumonia (VAP)) | hgcpoxdduh(jwzkwzzddg) = ywzadzyrdz wiupcfirjo (phxkkveeyn, qhsdvvuvph - cssvtxxafd) View more | ||||||
Phase 3 | 274 | baucrxlloo(oqrxijprku) = asdjceyflw kqqmglgeas (ggkkussomk, -5.0 to 18.5) View more | Negative | 13 Nov 2012 | |||
Imipenem-cilastatin | baucrxlloo(oqrxijprku) = mkrgppogmg kqqmglgeas (ggkkussomk ) View more | ||||||
Phase 4 | 30 | lryovoufoj(eivknmpfej) = crjwwvrhol hznqrasqbo (phnpqghkql, takeqcofpt - wnmkcuvoaq) View more | - | 25 Sep 2012 |