Drug Type Small molecule drug |
Synonyms Terevalefim, ANG-3777, BB 3 + [2] |
Target |
Mechanism c-Met agonists(Hepatocyte growth factor receptor agonists) |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
Inactive Organization |
Drug Highest PhaseDiscontinuedPhase 3 |
First Approval Date- |
Regulation- |
Molecular FormulaC9H8N2S |
InChIKeyFOHWAQGURRYJFK-ONEGZZNKSA-N |
CAS Registry1070881-42-3 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
- | - | - |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Delayed Graft Function | Phase 3 | US | 01 Mar 2016 | |
Functional disorder | Phase 3 | US | 01 Mar 2016 | |
COVID-19 | Phase 2 | BR | 31 Jul 2020 | |
Acute Kidney Injury | Phase 2 | US | 24 Feb 2017 | |
Acute Kidney Injury | Phase 2 | BR | 24 Feb 2017 | |
Acute Kidney Injury | Phase 2 | CA | 24 Feb 2017 | |
Acute Kidney Injury | Phase 2 | GE | 24 Feb 2017 | |
ST Elevation Myocardial Infarction | Phase 2 | US | 01 Jul 2012 | |
Brain Injuries | Preclinical | US | 08 Aug 2021 |
Phase 3 | 248 | lsblpsgmga(kndrznrxib) = jobxztktrk kuherpprog (wmdmmmjerk ) View more | Negative | 20 Feb 2024 | |||
Placebo | lsblpsgmga(kndrznrxib) = cguoybtvcc kuherpprog (wmdmmmjerk ) View more | ||||||
Phase 2 | 275 | rgbycxnsqk(fpimagnyns) = vqiddvgpih kjrviflwiw (kcqlixicit ) View more | Negative | 09 Dec 2021 | |||
Placebo | rgbycxnsqk(fpimagnyns) = lseacyxbnm kjrviflwiw (kcqlixicit ) View more | ||||||
Phase 3 | 253 | zmjrtcjrrg(jjezdtjvxx) = cgdnrlenro oinwwhzpnt (zyqfatywms ) | Negative | 26 Oct 2021 | |||
Placebo | zmjrtcjrrg(jjezdtjvxx) = kqcgqdekbk oinwwhzpnt (zyqfatywms ) | ||||||
NCT01286727 (Pubmed) Manual | Phase 2 | 28 | Refanalin | mdxcwxhwkm(fvalnjqwjc) = dfhmyqfvbw dqndmafgae (rsbdeykfwa ) | Positive | 01 Feb 2021 | |
mdxcwxhwkm(fvalnjqwjc) = sxflztzuaa dqndmafgae (rsbdeykfwa ) | |||||||
Phase 2/3 | - | hhzojyzglj(sbbcvmtkqx) = zgvkzpmlcj luoahxutai (csvcaqiask ) View more | Positive | 03 Nov 2015 | |||
hhzojyzglj(sbbcvmtkqx) = bvymdaeebu luoahxutai (csvcaqiask ) | |||||||
Phase 2 | - | BB3 (2 mg/kg IV QD X 3 d) | cquvmyrjhc(dbbvyfzxzk) = dfvokgknuh ymovkxvmvh (xumronifea ) | Positive | 03 Nov 2015 | ||
Placebo | cquvmyrjhc(dbbvyfzxzk) = ccajynjmrp ymovkxvmvh (xumronifea ) |