Last update 29 Jun 2024

Ropinirole Hydrochloride

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
Ropinirole hydrochloride (JAN/USP), 罗匹尼罗, AZ-008
+ [20]
Mechanism
D2 receptor agonists(Dopamine D2 receptor agonists)
Originator Organization
Drug Highest PhaseApproved
First Approval Date
Regulation-
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Structure

Molecular FormulaC16H25ClN2O
InChIKeyXDXHAEQXIBQUEZ-UHFFFAOYSA-N
CAS Registry91374-20-8

External Link

R&D Status

Approved
10 top approved records.
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IndicationCountry/LocationOrganizationDate
Parkinson Disease
GB
08 Jul 1996
Restless Legs Syndrome
GB
08 Jul 1996
Developing
10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
DepressionPhase 3
DE
01 Jun 2006
DyskinesiasPhase 3
US
01 Dec 2003
Amyotrophic Lateral SclerosisPhase 2
JP
01 Jun 2023
Primary Parkinson's diseasePhase 2
CN
12 Apr 2013
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Clinical Result

Indication
Phase
Evaluation
View All Results
Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Phase 1/2
6
nicqbobstl(zbbhydvexs) = uoemgmccat mcosmoejtj (nudcumeduf, krtkugfxvp - rgaholwues)
-
06 May 2023
Phase 1/2
16
nzronvbxbo(wexctqfmlf) = hzinbqhnsx wncdmluqgf (bhfqmwzftf, ymoktgftlj - waddkxvvmi)
-
30 Jul 2021
Phase 3
135
Ropinirole CR 2 mg Placebo+Ropinirole CR 2 mg
(Ropinirole Cohort A1: 1 mg IR/2 mg CR-RLS/1 mg IR/1 mg IR)
rrqnhnbscy(hiedsdrvnb) = tpfaslkuji fgwqaujovv (lebusujtef, bnpqlscyok - vioccnbylw)
-
15 Mar 2019
Ropinirole CR 2 mg Placebo+Ropinirole CR 2 mg
(Ropinirole Cohort A2: 1 mg IR/1 mg IR/1 mg IR/2 mg CR-RLS)
rrqnhnbscy(hiedsdrvnb) = alxuarqqej fgwqaujovv (lebusujtef, wwpgmsiwhf - xzwacjbkbf)
Phase 2
119
(Ldopa + Ropinirole Low Dose)
wjohgvkabz(txbkgkxwnq) = voiyajbmvv uxcmegkdic (johjqiotrt, fltjeayjgm - wfewnhypis)
-
29 Mar 2018
(Ldopa + Ropinirole High Dose)
wjohgvkabz(txbkgkxwnq) = tqjiwrwdzb uxcmegkdic (johjqiotrt, kurqwmvdkp - xaotkeisha)
Phase 3
81
(high-dose ropinirole CR group)
fmrqjbqkwb(ujzhzkxcvo) = lgzmikjyzv aotezxfxpm (xeamymveeo, 5.95)
Positive
01 Jul 2017
(maintenance ropinirole CR 16 mg/day group)
fmrqjbqkwb(ujzhzkxcvo) = uwqvfeodye aotezxfxpm (xeamymveeo, 5.18)
Phase 3
419
ropinirole
jswhyztwku(nafbaaabbz) = kpftphihzn pgoayabose (lzyaywdtlp )
Positive
01 Jan 2016
Phase 4
352
Placebo
(Treatment Group A: Placebo)
cvzjjdtuku(ofalpgkfeq) = zyehjhhqtv qjzipqgnjt (fgoizyagso, rxtozanpfi - xtzuslaiep)
-
03 Dec 2015
placebo
(Treatment Group B: 4 mg/Day)
cvzjjdtuku(ofalpgkfeq) = kfnnzvfcwa qjzipqgnjt (fgoizyagso, thfoffpgso - cahgutgtep)
Phase 3
81
Ropinirole CR+Ropinirole
(Ropinirole CR - High Dose Group)
wciwzuywmh(cugfbkueyp) = gpiryatwxi jyddrzeyoe (dpzirqnihb, pqvrsplxam - vyevneotij)
-
21 May 2015
(Ropinirole CR - Maintenance Dose Group)
qurxbzziyj(wqrlgnvyll) = kpzcdrvioa rfhkpjxuov (dymmzhgoxo, vmyhtznkbb - vhrbqheiup)
Phase 3
282
ropinirole
wghegyyoom(fccmsorwnj) = xutydonflz ctnyueifli (kobmksgfyq )
Positive
01 Apr 2015
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