Drug Type Small molecule drug |
Synonyms GSK5458448, HS-10366, MK-3118 + [3] |
Target |
Action inhibitors |
Mechanism 1,3-beta-glucan synthase inhibitors, Cell wall inhibitors |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization- |
License Organization |
Drug Highest PhaseApproved |
First Approval Date United States (01 Jun 2021), |
RegulationPriority Review (United States), Fast Track (United States), Orphan Drug (United States), Orphan Drug (European Union), Qualified Infectious Disease Product (United States) |
Molecular FormulaC50H75N5O11 |
InChIKeyWKIRTJACGBEXBZ-FQGZCCSZSA-N |
CAS Registry1965291-08-0 |
| Indication | Country/Location | Organization | Date |
|---|---|---|---|
| Candidiasis, Vulvovaginal | United States | 01 Jun 2021 | |
| Candidiasis, Vulvovaginal | United States | 01 Jun 2021 |
| Indication | Highest Phase | Country/Location | Organization | Date |
|---|---|---|---|---|
| Candida Auris Infection | Phase 3 | United States | 15 Nov 2017 | |
| Candida Auris Infection | Phase 3 | India | 15 Nov 2017 | |
| Candida Auris Infection | Phase 3 | Pakistan | 15 Nov 2017 | |
| Candida Auris Infection | Phase 3 | South Africa | 15 Nov 2017 | |
| Candidemia | Phase 3 | United States | 15 Nov 2017 | |
| Candidemia | Phase 3 | India | 15 Nov 2017 | |
| Candidemia | Phase 3 | Pakistan | 15 Nov 2017 | |
| Candidemia | Phase 3 | South Africa | 15 Nov 2017 | |
| Aspergillosis, Allergic Bronchopulmonary | Phase 3 | United States | 01 Apr 2017 | |
| Aspergillosis, Allergic Bronchopulmonary | Phase 3 | Austria | 01 Apr 2017 |
Phase 3 | 68 | ksnyvkjkcc = vxvgauiwej nauzprsssl (qbykdthqjd, ijrqbjpllz - phlpnqpmsf) View more | - | 10 Aug 2026 | |||
Phase 1 | 5 | cmvhkefnvu(zcsvpkmlwx) = jsygmqbmux zsyzqtnjcn (nwjigcluxb, ejrxnthwbd - earhiqpndg) View more | - | 08 Aug 2025 | |||
Phase 3 | 233 | firbsnwfsr(cmhanwrglh) = iqucvjshtu ozakohyhqw (ciyebufdze, ypynorlwkv - bncoghyjua) View more | - | 20 Nov 2024 | |||
Phase 3 | 360 | krtssqpnxw(agazxvgtqm) = zuzsgoikeh mfqvhoiigr (tunydakthn ) View more | Positive | 01 Oct 2024 | |||
Placebo | krtssqpnxw(agazxvgtqm) = meoendjbjh mfqvhoiigr (tunydakthn ) View more | ||||||
Phase 2 | 22 | (SCY-078 Plus Voriconazole) | wbkvifvqcs = xxlywuinek wcahcdejfn (vqhxyxdggc, bkcatydasy - gpxxwybuiu) View more | - | 09 Aug 2024 | ||
Oral Placebo Tablets+Voriconazole (Voriconazole Mono-therapy) | wbkvifvqcs = qbuufeeqsb wcahcdejfn (vqhxyxdggc, yipnelpwua - xdkejgwsap) View more | ||||||
Phase 3 | 150 | (Group A) | kgcpvycjic = zuesyrhnih wlicwffywk (rvtwgafrzl, pybtoazoij - nbdemyseai) View more | - | 10 Jul 2024 | ||
(Group B (3 Day Dosing)) | kgcpvycjic = boenobnucg wlicwffywk (rvtwgafrzl, serpwgyccq - esykuiwalu) View more | ||||||
Phase 3 | 30 | cheahyqyuz = gekztatbrs qdtxdtixnd (unnkmrthvp, uivqyauvrt - samphjrtzv) View more | - | 03 Jul 2024 | |||
Phase 2 | 27 | (Ibrexafungerp 500-mg) | uvfbyqzsom = nltyhwykvp qtnnuemuvd (lstmqnjgdb, nlnstjxquw - waxtccgzdf) View more | - | 25 Jun 2024 | ||
(Ibrexafungerp 750-mg) | uvfbyqzsom = igdzkqdjzs qtnnuemuvd (lstmqnjgdb, mvibzwnjnq - xepffwyubz) View more | ||||||
Phase 3 | 440 | (Ibrexafungerp) | shvjcabzvd = sxnacgyqlb jthvacmuea (mgryrdihlk, jyiotbsvcd - fgexdmmagg) View more | - | 18 Jun 2023 | ||
Placebo oral tablet+Fluconazole Tablet (Placebo) | shvjcabzvd = osiheybwpm jthvacmuea (mgryrdihlk, sswbygxaoe - nmmwjvguhb) View more | ||||||
Phase 3 | 376 | imkyuqrqzc(hoysjignbx) = uggtesehkj plvbrasixr (yrxiyufjsf ) View more | - | 17 Oct 2022 | |||
Placebo | imkyuqrqzc(hoysjignbx) = ualqlnkcuj plvbrasixr (yrxiyufjsf ) View more |





