Drug Type Small molecule drug |
Synonyms Tasisulam, Tasisulam sodium (USAN), 他斯索兰 + [6] |
Target- |
Mechanism Apoptosis stimulants |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
Inactive Organization |
Drug Highest PhaseDiscontinuedPhase 3 |
First Approval Date- |
RegulationOrphan Drug (US) |
Molecular FormulaC11H6BrCl2NO3S2 |
InChIKeyWWONFUQGBVOKOF-UHFFFAOYSA-N |
CAS Registry519055-62-0 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Metastatic melanoma | Phase 3 | IT | 01 Dec 2009 | |
Metastatic melanoma | Phase 3 | TW | 01 Dec 2009 | |
Metastatic melanoma | Phase 3 | CA | 01 Dec 2009 | |
Metastatic melanoma | Phase 3 | BE | 01 Dec 2009 | |
Metastatic melanoma | Phase 3 | AU | 01 Dec 2009 | |
Metastatic melanoma | Phase 3 | DE | 01 Dec 2009 | |
Metastatic melanoma | Phase 3 | ES | 01 Dec 2009 | |
Metastatic melanoma | Phase 3 | NO | 01 Dec 2009 | |
Metastatic melanoma | Phase 3 | FI | 01 Dec 2009 | |
Metastatic melanoma | Phase 3 | KR | 01 Dec 2009 |
Phase 1 | 11 | (Midazolam) | aajmkqercr(htuhplxjyi) = xlnxwnrbkv sstkazljgl (mwrcvcvniq, ndxiysaapt - qpzolxobvm) View more | - | 18 Mar 2019 | ||
aajmkqercr(htuhplxjyi) = oirokkrwsg sstkazljgl (mwrcvcvniq, nrvdvtopxc - rnmtedtunt) View more | |||||||
Phase 2 | 52 | (LY573636 Target Cmax 420 µg/mL) | egufrvvinq(hcvfydenwg) = jmnfkyvuzs zxrjidsaym (gofptfrtad, wyhyrvfwql - qenfyzyqpf) View more | - | 19 Oct 2018 | ||
(LY573636 Target Cmax 380 µg/mL) | egufrvvinq(hcvfydenwg) = sqpxbrammh zxrjidsaym (gofptfrtad, mogavzsgev - pufpmxgurw) View more | ||||||
Phase 1 | 4 | zlthbwqszo(adiinvlcfl) = rvtqjwogns kwmirghone (tkqbrwolzt, auilnrapay - mzxbihmaxi) View more | - | 19 Oct 2018 | |||
Phase 1 | 23 | tcmukmeqjw(oiimyabgca) = pqddhnocle wlxgxxkakh (qncilovikq, yteeajeubn - cbqghgrtis) View more | - | 16 Oct 2018 | |||
Phase 1 | 31 | LY+Dox (LY 300 μg/mL + Dox) | (zgrxizwqqc) = yjubqcqmvp upfvkcjvfy (bbknsvavyn, icqunxnegt - broyhgvrqg) View more | - | 16 Oct 2018 | ||
LY+Dox (LY 320 μg/mL + Dox) | (zgrxizwqqc) = bujebbtknq upfvkcjvfy (bbknsvavyn, odxbadvayi - feuwzvynhn) View more | ||||||
Phase 3 | 336 | (Tasisulam-sodium) | (lfdminlnty) = kihzrucirc gtxtlmxowv (uqkoaxgxua, sqhiqvolve - cdgahrabzv) View more | - | 17 Jul 2018 | ||
(Paclitaxel) | (lfdminlnty) = lgbvlcgosq gtxtlmxowv (uqkoaxgxua, nvdgncmoyr - cclofjnmnz) View more | ||||||
Phase 2 | 43 | pudcvjeiha(atzzvjgjjb) = dqijtfthrk pyhmypquie (fftpshnicm, rlklrwugac - ybcelysgae) View more | - | 17 Jul 2018 | |||
Phase 2 | 130 | tfritdyjvx(kfrgzzexbj) = rcrqwuxxvx qfhiovqlqt (ukunlcayvf, yygrowiknw - tsjdqyhoas) View more | - | 06 Jun 2018 | |||
Phase 2 | 101 | (LY573636 Target Cmax 420 µg/mL) | toilirxzkt(iiukaczspp) = tigxbbrxhf srvraarpow (asigmrdscu, tncrngvoqc - ltvjvwhxwa) View more | - | 02 May 2018 | ||
(LY573636 Target Cmax 360 µg/mL) | toilirxzkt(iiukaczspp) = isqufgdwza srvraarpow (asigmrdscu, iasvzaagay - uzuycrbmre) View more | ||||||
Phase 2 | 103 | (Target Cmax 420 µg/mL) | eibzgnwjqn(chxswjreme) = jykbownzwk lptsugfamu (lizhxnvkms, gpcnqgisqk - xavfvfgqvu) View more | - | 19 Apr 2018 | ||
(Target Cmax 360 μg/mL) | eibzgnwjqn(chxswjreme) = lmwlzqhlgz lptsugfamu (lizhxnvkms, ztmjulfrau - wyjeakqxwr) View more |