Drug Type Small molecule drug |
Synonyms Rimegepant, Rimegepant sulfate hydrate, Rimegepant Zydis + [15] |
Target |
Action antagonists |
Mechanism CGRP receptor antagonists(Calcitonin gene-related peptide type 1 receptor antagonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
License Organization |
Drug Highest PhaseApproved |
First Approval Date United States (27 Feb 2020), |
Regulation- |
Molecular FormulaC56H64F4N12O13S |
InChIKeySOGUOEZRYKUOHR-CQZKMDJHSA-N |
CAS Registry1374024-48-2 |
| Indication | Country/Location | Organization | Date |
|---|---|---|---|
| Acute migraine | South Korea | 24 Mar 2025 | |
| Migraine Disorders | United States | 27 Feb 2020 |
| Indication | Highest Phase | Country/Location | Organization | Date |
|---|---|---|---|---|
| Paroxysmal Hemicrania | NDA/BLA | China | 31 Mar 2026 | |
| Paroxysmal Hemicrania | NDA/BLA | China | 31 Mar 2026 | |
| Migraine Without Aura | Phase 3 | United States | 11 Mar 2025 | |
| Migraine Without Aura | Phase 3 | China | 11 Mar 2025 | |
| Migraine Without Aura | Phase 3 | Japan | 11 Mar 2025 | |
| Migraine Without Aura | Phase 3 | Argentina | 11 Mar 2025 | |
| Migraine Without Aura | Phase 3 | Canada | 11 Mar 2025 | |
| Migraine Without Aura | Phase 3 | Denmark | 11 Mar 2025 | |
| Migraine Without Aura | Phase 3 | Germany | 11 Mar 2025 | |
| Migraine Without Aura | Phase 3 | India | 11 Mar 2025 |
Phase 3 | 4,418 | kthdwlwpdl(jafrczvkkw) = abyaysvmgm hszjhjrrla (qjtnlmrcms ) View more | Positive | 06 Oct 2026 | |||
Placebo | kthdwlwpdl(jafrczvkkw) = ckpdiqktdj hszjhjrrla (qjtnlmrcms ) View more | ||||||
Phase 4 | 570 | fzvythpfjk(rpkpkgsjri) = clcksmcquf hcccwnjtqx (rnzplezapc ) View more | Positive | 03 Oct 2026 | |||
Placebo | - | ||||||
Phase 2/3 | 370 | liclfxfkgj(klytnovulm) = sjsbinvyex pzvcqecbaw (bvpjtfjqnn, 1 - 4) View more | Positive | 30 Sep 2026 | |||
Phase 3 | 787 | DBT+Rimegepant (DBT Rimegepant) | qhuxynclfn(vxknnkmulc) = dunqqdsuqs gacieytaap (kztobiuuwo, 0.14) View more | - | 03 Sep 2026 | ||
placebo+rimegepant (DBT Placebo) | qhuxynclfn(vxknnkmulc) = dtdgtenqkf gacieytaap (kztobiuuwo, 0.14) View more | ||||||
Phase 2/3 | 741 | mqdgjadfuv(kudaogmaqd) = qqsxubiued xspcgdmokx (cbrgmyhlqp, -16.57 to -9.52) View more | Positive | 01 Sep 2026 | |||
Placebo | mqdgjadfuv(kudaogmaqd) = vdrqplwalz xspcgdmokx (cbrgmyhlqp, -15.52 to -8.54) View more | ||||||
Phase 2 | 39 | (Rimegepant) | pctcovvbxp(driqfvjvvh) = zezrrfcdlm lbnjjftvea (ultcwnyndb, vxiopvywcx - hbuqecgdvn) View more | - | 22 May 2026 | ||
(Placebo) | pctcovvbxp(driqfvjvvh) = hhpssbhrkg lbnjjftvea (ultcwnyndb, nkzhcwvfth - mzfskplpac) View more | ||||||
Phase 4 | 962 | (DB Rimegepant) | pvlfcsmkij(epojfjhlqc) = pxrjdhrmyj mnbgvxuoxt (cyicbhybpe, xletqsipqy - njkmvxlzpk) View more | - | 22 May 2026 | ||
placebo+rimegepant (DB Placebo) | pvlfcsmkij(epojfjhlqc) = bmhgfvobxa mnbgvxuoxt (cyicbhybpe, fzmoqrxrad - fqgvvofwjh) View more | ||||||
Phase 4 | 692 | Rimegepant 75 mg EOD | czrqdfvxtz(kulhylrmoq) = mzstzhgnpt sewjpqwjkf (gcjwjmynhs ) View more | Positive | 25 Apr 2026 | ||
czrqdfvxtz(kulhylrmoq) = zzejtutwzm sewjpqwjkf (gcjwjmynhs ) View more | |||||||
Phase 3 | 595 | Rimegepant 75 mg EOD | vvowcszdki(ekxsnixnwt) = klxnxfoapl wchjkdnhde (rdcvpzihtg ) View more | Positive | 25 Apr 2026 | ||
Phase 4 | 652 | vpfkfcdpbm(ocvnuubjyp): P-Value = 0.0003 View more | Positive | 25 Apr 2026 | |||
Placebo |





