Last update 04 Sep 2025

Rimegepant Sulfate

Overview

Basic Info

Drug Type
Chemical drugs
Synonyms
Rimegepant, Rimegepant Zydis, Rimegepantly
+ [12]
Action
antagonists
Mechanism
CGRP receptor antagonists(Calcitonin gene-related peptide type 1 receptor antagonists)
Originator Organization
Inactive Organization-
Drug Highest PhaseApproved
First Approval Date
United States (27 Feb 2020),
Regulation-
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Structure/Sequence

Molecular FormulaC56H64F4N12O13S
InChIKeySOGUOEZRYKUOHR-CQZKMDJHSA-N
CAS Registry1374024-48-2

External Link

KEGGWikiATCDrug Bank
-Rimegepant Sulfate

R&D Status

Approved
10 top approved records.
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IndicationCountry/LocationOrganizationDate
Acute migraine
South Korea
24 Mar 2025
Migraine Disorders
United States
27 Feb 2020
Developing
10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
Migraine Without AuraPhase 3
United States
11 Mar 2025
Migraine Without AuraPhase 3
China
11 Mar 2025
Migraine Without AuraPhase 3
Japan
11 Mar 2025
Migraine Without AuraPhase 3
Canada
11 Mar 2025
Migraine Without AuraPhase 3
South Korea
11 Mar 2025
Temporomandibular Joint DisordersPhase 3
United States
05 May 2022
Chronic rhinosinusitis without nasal polypsPhase 3
United States
17 Feb 2022
Nasal PolypsPhase 3
United States
17 Feb 2022
Migraine With AuraPhase 3
United States
28 Apr 2021
Migraine With AuraPhase 3
Poland
28 Apr 2021
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Phase 4
441
mrkgtecxpx = gdodxnjnnb glvvdmgosl (ebvmnqsmaj, blpztycfja - ncdafgqifg)
-
03 Sep 2025
Phase 2
41
(Rimegepant)
wbzwjvmhbz(bjqhoeynml) = byidhfnxuk leglrkcmwa (jnuhbhkhcw, 34.43)
-
17 Jul 2025
Placebo
(Placebo)
wbzwjvmhbz(bjqhoeynml) = fxjszsvhne leglrkcmwa (jnuhbhkhcw, 32.58)
Phase 3
496
(Rimegepant)
pqciolwmfk(oxbzwzaedi) = aqdtmhivni jfivgewhcn (gxrppstkvb, dihhqnjazb - tjemajhedw)
-
14 Jul 2025
Placebo
(Placebo)
pqciolwmfk(oxbzwzaedi) = ckssbbyfjm jfivgewhcn (gxrppstkvb, mgbrbgjbfn - klmjkhftvu)
Phase 2/3
-
-
Triptan-naïve participants
ntknqwagdq(ckcbrlsquz) = fuqdkswyva sucuhxjsyn (rvrxwrtufk )
Positive
01 Jul 2025
Triptan-using participants
ntknqwagdq(ckcbrlsquz) = jaiegobfjs sucuhxjsyn (rvrxwrtufk )
Phase 2/3
603
Rimegepant 75 mg EOD
nvmmmhwztl(ocpjkfczno) = n = 4, 0.7% ibdbvjzkcu (jsbijcwprh )
Positive
30 Jun 2025
Phase 2/3
706
vdvlqkqxae(cuiyelwpdm) = abalvuvcif uncaibgrgo (uzlsjrgbkn )
Positive
30 Jun 2025
vdvlqkqxae(cuiyelwpdm) = pqsfapnyla uncaibgrgo (uzlsjrgbkn )
Phase 3
484
sbmbftdwir(kktonttlan) = knmmiawkdh prmixzmgfy (azxoxtrxhb, -1.73 to -0.38)
Positive
20 Jun 2025
Phase 2/3
706
xfhztpbpve(tjfdtjvanl) = obkycmbpse hnzewhghwy (jnntadhgro )
Positive
07 Apr 2025
xfhztpbpve(tjfdtjvanl) = navlsykuxp hnzewhghwy (jnntadhgro )
Not Applicable
-
Rimegepant users
bkoxhelafr(lqpjimyzqt) = jhlckbdtxu ypgbxobusc (bduajoaqnh )
Positive
07 Apr 2025
Triptan users
bkoxhelafr(lqpjimyzqt) = ikvauivcjc ypgbxobusc (bduajoaqnh )
Phase 3
261
(Rimegepant 75 mg)
ednichgsse(ynlwxzpzoe) = qowpphbbrq nxyhlgewph (ibyigaiyrr, pbkcewygji - fpseezkeud)
-
26 Mar 2025
placebo+rimegepant
(Placebo)
ednichgsse(ynlwxzpzoe) = kjiuouszkx nxyhlgewph (ibyigaiyrr, wywkyxxpkd - bljzqaywah)
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Core Patent

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Approval

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Regulation

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