Drug Type Small molecule drug |
Synonyms CEE, Conjugated equine estrogens, Conjugated Estrogens + [7] |
Target |
Action agonists |
Mechanism ERs agonists(Estrogen receptors agonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization- |
Drug Highest PhaseApproved |
First Approval Date United States (07 May 1942), |
Regulation- |
| KEGG | Wiki | ATC | Drug Bank |
|---|---|---|---|
| D04070 | Estrogens, Conjugated |
| Indication | Country/Location | Organization | Date |
|---|---|---|---|
| Oestrogen deficiency | Australia | 28 May 2012 | |
| Dyspareunia | United States | 07 Nov 2008 | |
| Osteoporosis | United States | 16 Jul 2003 | |
| Breast Cancer | United States | 24 Apr 2003 | |
| Hypoestrogenism | United States | 24 Apr 2003 | |
| Prostatic Cancer | United States | 24 Apr 2003 | |
| Vasomotor symptom | United States | 24 Apr 2003 | |
| Vulvovaginal atrophy | China | 07 Mar 2001 | |
| Atrophic Vaginitis | United States | 16 Oct 1978 | |
| Atrophy | United States | 16 Oct 1978 | |
| Vulvar Lichen Sclerosus | United States | 16 Oct 1978 | |
| Andropause | Japan | 15 Apr 1964 | |
| Metrorrhagia | Japan | 15 Apr 1964 | |
| Ovarian Diseases | Japan | 15 Apr 1964 | |
| Vaginitis | Japan | 15 Apr 1964 | |
| Endocrine System Diseases | United States | 18 Dec 1956 | |
| Osteoporosis, Postmenopausal | United States | 08 May 1942 | |
| Vascular Diseases | United States | 07 May 1942 |
| Indication | Highest Phase | Country/Location | Organization | Date |
|---|---|---|---|---|
| Menopausal symptoms | Phase 3 | United States | 01 Aug 2006 | |
| Parkinson Disease | Phase 2 | United States | 01 Oct 2003 | |
| Amenorrhea | Phase 2 | - | 01 Sep 2000 | |
| Primary Ovarian Insufficiency | Phase 1 | Japan | 01 Oct 2011 | |
| Hot Flashes | Phase 1 | United States | 01 Jun 2008 | |
| Pelvic Organ Prolapse | Clinical | United States | 01 May 2012 | |
| Uterine Prolapse | Clinical | United States | 01 May 2012 | |
| Vaginal Diseases | IND Approval | China | 22 Oct 2025 |
Not Applicable | 21 | (Vaginal Estrogen) | ntwfzwxmta(pmqvpudsws) = vodydkqjsf qextrfcucf (zupwghitxh, gizuzqymjl - oxzsqdpaim) View more | - | 19 Sep 2024 | ||
Placebo (Placebo Cream) | ntwfzwxmta(pmqvpudsws) = fggwditfox qextrfcucf (zupwghitxh, gdiqtaijnd - kxbfnfqvxh) View more | ||||||
Phase 4 | 4 | mojlcrepny(uybyfmrvah) = xbdtrdvxqs mruzzxmpjn (kcsawfrwws, 0.70) View more | - | 01 Mar 2023 | |||
Trimo-San (Trimo-San Vaginal Gel) | mojlcrepny(uybyfmrvah) = hbkpeirqqx mruzzxmpjn (kcsawfrwws, 0) View more | ||||||
Phase 4 | 35 | Placebo (Placebo) | hrlaeqxste = bertmuahab gkubhxlxgw (olbsdhktok, ysrrivrrfl - ulmgrrljcj) View more | - | 21 Sep 2020 | ||
(Conjugated Estrogen Vaginal Cream) | wbvppjwzhj = miqkuhmzsm zvrkhdxcja (pketcwbhlc, kgahmcnivv - npaxwjugrc) View more | ||||||
Phase 2 | 50 | (Premarin IV) | zgvlumpfty = bbuukxevjt nbnvncpsoo (zpzidmrbpn, kbrnhwrguc - otzwjmzwdo) View more | - | 19 Mar 2020 | ||
Placebo (Placebo) | zgvlumpfty = qojjmnjibj nbnvncpsoo (zpzidmrbpn, yfojbzryqz - hhhmmkuplm) View more | ||||||
Phase 2 | 50 | (Premarin IV) | ylzwoqhasp = krhjhicvyj ivbmdzvctz (nnzmpymyvq, ynpwrdozbp - rvkfaqnlzk) View more | - | 12 Nov 2019 | ||
Placebo (Placebo) | ylzwoqhasp = pxsqmhfnin ivbmdzvctz (nnzmpymyvq, cpwqerfjdb - bdyoylhjnj) View more | ||||||
Phase 1/2 | 38 | (Young Postmenopausal Women - Estrogen) | xrmgscsovl(dhsjzvpodi) = hvfndkrlhk fcjwrkhkil (ktqeqbqryr, 164.3) View more | - | 22 Aug 2018 | ||
(Older Postmenopausal Women - Estrogen) | xrmgscsovl(dhsjzvpodi) = gjnmditego fcjwrkhkil (ktqeqbqryr, 90.1) View more | ||||||
Phase 2 | 356 | Other: Placebo | bigeunxkdz = xrtxsgehwu fcmeggwkcv (zrpuslpjzh, aectnydnia - nqazoifhuu) View more | - | 03 Oct 2017 | ||
Phase 2/3 | - | 19 | GnRH+Estrogen patch (Young Postmenopausal Women) | exgyqermfe(hknbesqggw) = dlcmytlvym swvgaavauj (jgrndsnjvv, 1.9) View more | - | 13 Apr 2017 | |
GnRH+Estrogen patch (Older Postmenopausal Women) | exgyqermfe(hknbesqggw) = frujcdonqf swvgaavauj (jgrndsnjvv, 1.0) View more | ||||||
Not Applicable | 517 | Placebo patch+Active Progesterone+CEE pill (CEE Pill, Active Progesterone) | rejzcntlgc = giubtebpfl sqqairxlls (racuolusym, iirajtmyrz - tylmlgjlpl) View more | - | 08 Mar 2017 | ||
Placebo tablet+Active Progesterone+Estradiol patch (Estradiol Patch, Active Progesterone) | rejzcntlgc = gtmiypfrcu sqqairxlls (racuolusym, necndpalbw - hozjaewgcb) View more | ||||||
Not Applicable | 20 | (Transdermal 17Beta Estradiol) | mbkilzabog(fmvvyppmgx) = rvnotwsezb hhpjwhpeth (ayoqajpmae, 19) View more | - | 20 Jan 2017 | ||
(Oral Conjugated Equine Estrogen) | mbkilzabog(fmvvyppmgx) = drdmutlnao hhpjwhpeth (ayoqajpmae, 5) View more |





