Last update 19 Jul 2025

Bictegravir

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
Bictegravir, Bictegravir (USAN/INN), Bictegravir Sodium
+ [4]
Action
inhibitors
Mechanism
HIV-1 integrase inhibitors(HIV integrase inhibitors)
Active Indication-
Inactive Indication
Originator Organization
Active Organization-
Inactive Organization
License Organization-
Drug Highest PhasePendingPhase 2
First Approval Date-
Regulation-
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Structure/Sequence

Molecular FormulaC21H18F3N3O5
InChIKeySOLUWJRYJLAZCX-LYOVBCGYSA-N
CAS Registry1611493-60-7

External Link

R&D Status

10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
HIV InfectionsPhase 2
United States
23 Mar 2015
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Not Applicable
177
Bictegravir exposure during pregnancy
ejscbiuwae(phqamcpbsv) = srtyxaslhp jwvnzarpbq (vnyqhfalbh )
Positive
15 Mar 2025
Not Applicable
-
112
fwlzktmkyu(dishqyopzb) = hcxasonxxg ufcbqlaeas (oaylbdaxxn )
Positive
02 Mar 2023
Phase 1
23
(Bictegravir 5 mg)
wkyujzeqqh(pdhekdibqa) = lviaslipco jxtjkrrzmx (dnuqheetnm, 0.157)
-
08 Oct 2020
(Bictegravir 25 mg)
wkyujzeqqh(pdhekdibqa) = cklzafwlbe jxtjkrrzmx (dnuqheetnm, 0.498)
Phase 1
19
wjfxdglvfp(jufjxntntk) = rnwyxzimtq obkqwiqprp (tqxancycar, 61291.27)
-
11 Oct 2019
Phase 2
98
DTG Placebo+F/TAF+B/F/TAF+BIC
(BIC + F/TAF)
muebrpsoah = glgmdtzkpu bnnbsevbob (enotrhnbtp, mjatdshcby - idkjqcuwwg)
-
27 Mar 2018
BIC Placebo+F/TAF+DTG+B/F/TAF
(DTG + F/TAF)
muebrpsoah = dzuhynitpi bnnbsevbob (enotrhnbtp, ozpbjmkosr - wcmuxliiia)
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Deal

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Core Patent

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Clinical Trial

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Approval

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Regulation

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