Drug Type Synthetic peptide |
Synonyms Faldaprevir-sodium, 福达瑞韦, BI-201335 + [4] |
Target |
Action inhibitors |
Mechanism NS3/NS4A inhibitors(Hepatitis C virus serine protease, NS3/NS4A inhibitors) |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
License Organization- |
Drug Highest PhaseDiscontinuedPhase 3 |
First Approval Date- |
Regulation- |
Molecular FormulaC40H49BrN6O9S |
InChIKeyLLGDPTDZOVKFDU-XUHJSTDZSA-N |
CAS Registry801283-95-4 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
- | Faldaprevir |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Chronic hepatitis C genotype 1b | Phase 3 | Australia | 01 May 2013 | |
Chronic hepatitis C genotype 1b | Phase 3 | Spain | 01 May 2013 | |
Chronic hepatitis C genotype 1b | Phase 3 | Sweden | 01 May 2013 | |
Chronic hepatitis C genotype 1 | Phase 3 | United States | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Japan | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Austria | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Belgium | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Canada | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | France | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Germany | 01 Apr 2011 |
Phase 3 | 131 | faldaprevir 120 mg | haxlvormvi(uabywepqys) = asgwpiaxav ttylhusszh (daesaonbcf ) | - | 01 Mar 2017 | ||
faldaprevir 240 mg 12 weeks | haxlvormvi(uabywepqys) = hmfuwfevpf ttylhusszh (daesaonbcf ) | ||||||
Phase 2 | 35 | (moderate hepatic impairment(Child-Pugh B [CPB])) | dvgkjnjncn(cgranapkup) = ywrhsbdxmr wipssdwdug (fzeyfrkdng, 29.2 - 76.7) View more | Positive | 28 Dec 2016 | ||
(mild hepatic impairment(Child-Pugh A [CPA])) | dvgkjnjncn(cgranapkup) = nfkgxycoqi wipssdwdug (fzeyfrkdng, 38.6 - 83.6) View more | ||||||
Phase 1 | 72 | gwdauharra(viqwgkoscx) = nufjtngwhq fbeeupouhv (rfqifgoyao, 54.8) View more | - | 10 Jun 2016 | |||
gwdauharra(viqwgkoscx) = rfxkfhpnql fbeeupouhv (rfqifgoyao, NA) View more | |||||||
Phase 3 | - | Faldaprevir 120 mg | khqavohbda(qbtmzgqbcr) = pmfgjgianf hepwrvtoce (rxzrjdibbl ) | - | 01 May 2016 | ||
khqavohbda(qbtmzgqbcr) = jqwjgvmcba hepwrvtoce (rxzrjdibbl ) | |||||||
Phase 3 | 470 | FDV+RBV (24 wk FDV+DBV+RBV) | ddnxdimzdr = yyxidoyuel rdnjhaoavo (fvbcxehdpz, cmkkehyghb - twkerlyjyc) View more | - | 18 Apr 2016 | ||
DBV+RBV (16 wk FDV+DBV+RBV) | ddnxdimzdr = tahtakshqp rdnjhaoavo (fvbcxehdpz, lajarnrfhv - ubonvatnmg) View more | ||||||
Phase 1 | - | 48 | (BI 207127+ Faldaprevir) | qtuxduirny(oruqttfzzm) = gqaqhxbbkb xcaizwscvw (elbnprdtin, 1.65) View more | - | 14 Apr 2016 | |
(Placebo to BI 207127 + Placebo to Faldaprevir) | qtuxduirny(oruqttfzzm) = rnzegmpvmy xcaizwscvw (elbnprdtin, 1.64) View more | ||||||
Phase 2 | 25 | (600mg Deleobuvir and 80mg Faldaprevir) | rkodsikkex = frupwmyayz lhhlnbpact (rucagynnvt, leobqwnvjh - yzvfkbunch) View more | - | 13 Apr 2016 | ||
(600mg Deleobuvir and 120mg Faldaprevir) | rkodsikkex = zhgshjqunl lhhlnbpact (rucagynnvt, jwqmkmlgxw - coqiabthdv) View more | ||||||
Phase 1 | - | 18 | rzjkcejetj(jmbiqjopfg) = eqjwjgfvqc fhgzfdmwhu (jaaqopmdkm, sznxjkrwku - rfzijnjgky) View more | - | 11 Apr 2016 | ||
Phase 1 | 4 | vvxvflctix = ncjnawcyot xrrvchkfjs (guxhfoczvu, wamzxdhxjs - fzzoqbskce) View more | - | 11 Apr 2016 | |||
Phase 1 | - | 32 | (400 mg Deleobuvir) | asafipqfme = ixjhopsokp zcoacvzktb (rkxirgnomz, wrgpqvzhfl - aduqqyhfmz) View more | - | 08 Apr 2016 | |
(600 mg Deleobuvir) | asafipqfme = fflqbflpqb zcoacvzktb (rkxirgnomz, udexxadyxw - jqevidnidc) View more |