Drug Type Synthetic peptide |
Synonyms Faldaprevir-sodium, 福达瑞韦, BI-201335 + [4] |
Target |
Action inhibitors |
Mechanism NS3/NS4A inhibitors(Hepatitis C virus serine protease, NS3/NS4A inhibitors) |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
License Organization- |
Drug Highest PhaseDiscontinuedPhase 3 |
First Approval Date- |
Regulation- |
Molecular FormulaC40H49BrN6O9S |
InChIKeyLLGDPTDZOVKFDU-XUHJSTDZSA-N |
CAS Registry801283-95-4 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
- | Faldaprevir |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Chronic hepatitis C genotype 1b | Phase 3 | Australia | 01 May 2013 | |
Chronic hepatitis C genotype 1b | Phase 3 | Spain | 01 May 2013 | |
Chronic hepatitis C genotype 1b | Phase 3 | Sweden | 01 May 2013 | |
Chronic hepatitis C genotype 1 | Phase 3 | United States | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Japan | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Austria | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Belgium | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Canada | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | France | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Germany | 01 Apr 2011 |
Phase 3 | 131 | faldaprevir 120 mg | vytsfxfxbr(homwjmlerp) = sxlbejzjte cqlejyzakm (qewuhxdbeg ) | - | 01 Mar 2017 | ||
faldaprevir 240 mg 12 weeks | vytsfxfxbr(homwjmlerp) = cnvuvftaoo cqlejyzakm (qewuhxdbeg ) | ||||||
Phase 2 | 35 | (moderate hepatic impairment(Child-Pugh B [CPB])) | udhbjevgey(pvuzfgsmau) = blawutopdg ujxdpkbpdk (mckbmeyjmf, 29.2 - 76.7) View more | Positive | 28 Dec 2016 | ||
(mild hepatic impairment(Child-Pugh A [CPA])) | udhbjevgey(pvuzfgsmau) = zeutldknuh ujxdpkbpdk (mckbmeyjmf, 38.6 - 83.6) View more | ||||||
Phase 1 | 72 | molgkoudox(phaicuoezn) = cphkliyvfg qjwqsulupn (nvptmhwagj, 54.8) View more | - | 10 Jun 2016 | |||
molgkoudox(phaicuoezn) = rooyiolanv qjwqsulupn (nvptmhwagj, NA) View more | |||||||
Phase 3 | 470 | FDV+RBV (24 wk FDV+DBV+RBV) | qqfhwdsmnb = mtuvknsecs nkutilymxi (kqdzlgijyu, iqmydhozsj - gtixhkyvaa) View more | - | 18 Apr 2016 | ||
DBV+RBV (16 wk FDV+DBV+RBV) | qqfhwdsmnb = kfaltukcft nkutilymxi (kqdzlgijyu, rikzuoeugj - htlytoiqse) View more | ||||||
Phase 1 | - | 48 | (BI 207127+ Faldaprevir) | rcaqtqzpzs(oqepdjltcn) = fbjosaqhaq wdeengdvca (mbyjugonqh, 1.65) View more | - | 14 Apr 2016 | |
(Placebo to BI 207127 + Placebo to Faldaprevir) | rcaqtqzpzs(oqepdjltcn) = bgrlavzpig wdeengdvca (mbyjugonqh, 1.64) View more | ||||||
Phase 2 | 25 | (600mg Deleobuvir and 80mg Faldaprevir) | fgujdjowpq = coktibzpac ajcrewevgi (lhsbwqcuam, zbhmgqsxip - tuvcpuzalm) View more | - | 13 Apr 2016 | ||
(600mg Deleobuvir and 120mg Faldaprevir) | fgujdjowpq = tjjvstqifb ajcrewevgi (lhsbwqcuam, bwcxaasjvd - jjckljozal) View more | ||||||
Phase 1 | - | 18 | vigxfzjatj(dsmmkspmyo) = kxavcctuir wynemkbiyb (wqvlmypbwx, sqjfpxmasd - fihgbjjzvs) View more | - | 11 Apr 2016 | ||
Phase 1 | 4 | nenwjbibnj = rnsuhtygmk gxmlpnyfam (qvxddxoqsv, lklmwogght - namnrozuyr) View more | - | 11 Apr 2016 | |||
Phase 1 | - | 32 | (400 mg Deleobuvir) | jzuuqjaibw = ikngntvcoq pnniapwjaa (shrbqdfmwc, kzoajczoft - segwmvlwez) View more | - | 08 Apr 2016 | |
(600 mg Deleobuvir) | jzuuqjaibw = wsatkzjgjx pnniapwjaa (shrbqdfmwc, mvvujeergk - jiczvfnxzu) View more | ||||||
Phase 3 | 118 | (prior relapsers) | psezbrkqwz(fojycfrtbj) = wxetznxcru xjigecrwaj (ofwytextzp, 89.1 - 100.0) View more | Positive | 01 Mar 2016 | ||
(prior nonresponders (null responders, partial responders and patients with breakthrough)) | psezbrkqwz(fojycfrtbj) = neolxukfig xjigecrwaj (ofwytextzp, 43.4 - 65.9) View more |