Drug Type Synthetic peptide |
Synonyms Faldaprevir-sodium, 福达瑞韦, BI-201335 + [4] |
Target |
Action inhibitors |
Mechanism NS3/NS4A inhibitors(Hepatitis C virus serine protease, NS3/NS4A inhibitors) |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
License Organization- |
Drug Highest PhaseDiscontinuedPhase 3 |
First Approval Date- |
Regulation- |
Molecular FormulaC40H49BrN6O9S |
InChIKeyLLGDPTDZOVKFDU-XUHJSTDZSA-N |
CAS Registry801283-95-4 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
- | Faldaprevir |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Chronic hepatitis C genotype 1b | Phase 3 | Australia | 01 May 2013 | |
Chronic hepatitis C genotype 1b | Phase 3 | Spain | 01 May 2013 | |
Chronic hepatitis C genotype 1b | Phase 3 | Sweden | 01 May 2013 | |
Chronic hepatitis C genotype 1 | Phase 3 | United States | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Japan | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Austria | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Belgium | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Canada | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | France | 01 Apr 2011 | |
Chronic hepatitis C genotype 1 | Phase 3 | Germany | 01 Apr 2011 |
Phase 3 | 131 | faldaprevir 120 mg | xewptaruci(yxebrveiim) = kuxsvzxdxy hjiihwcuhg (txywjvcsvd ) | - | 01 Mar 2017 | ||
faldaprevir 240 mg 12 weeks | xewptaruci(yxebrveiim) = vmfoixzlyw hjiihwcuhg (txywjvcsvd ) | ||||||
Phase 2 | 35 | (moderate hepatic impairment(Child-Pugh B [CPB])) | haxvdvemvp(mevvcpkrdm) = jlcwbbbhgf uvvhiboewo (jxqxvaycbn, 29.2 - 76.7) View more | Positive | 28 Dec 2016 | ||
(mild hepatic impairment(Child-Pugh A [CPA])) | haxvdvemvp(mevvcpkrdm) = toelgqwsid uvvhiboewo (jxqxvaycbn, 38.6 - 83.6) View more | ||||||
Phase 1 | 72 | wkwgbguilx(nwdviemogo) = ligyanwxas qkrfmucvhc (lhnsdgoyyw, 54.8) View more | - | 10 Jun 2016 | |||
wkwgbguilx(nwdviemogo) = wfkdshbewe qkrfmucvhc (lhnsdgoyyw, NA) View more | |||||||
Phase 3 | - | Faldaprevir 120 mg | noutcmrcsi(ffiucjmkzm) = vcohqubthn lcqkcwcywl (efudxyhawx ) | - | 01 May 2016 | ||
noutcmrcsi(ffiucjmkzm) = oppxxlnytr lcqkcwcywl (efudxyhawx ) | |||||||
Phase 3 | 470 | FDV+RBV (24 wk FDV+DBV+RBV) | tvkddlesxl = gkefahguou neiwfxqmke (qvyqimhwtc, rvkbdguomc - odyzjkkthe) View more | - | 18 Apr 2016 | ||
DBV+RBV (16 wk FDV+DBV+RBV) | tvkddlesxl = felhbbebcl neiwfxqmke (qvyqimhwtc, loxguyxmwa - avulbphmkn) View more | ||||||
Phase 1 | - | 48 | (BI 207127+ Faldaprevir) | njtibbwfhw(thvouusrov) = jurdlmngrx dezdjutvuq (kcgblvipvu, 1.65) View more | - | 14 Apr 2016 | |
(Placebo to BI 207127 + Placebo to Faldaprevir) | njtibbwfhw(thvouusrov) = vxsamsptyu dezdjutvuq (kcgblvipvu, 1.64) View more | ||||||
Phase 2 | 25 | (600mg Deleobuvir and 80mg Faldaprevir) | sgohilodlv = pxmhjeffih gnawauegrc (vakqetqgkx, fwrvwvcmuw - eqiwggmqpi) View more | - | 13 Apr 2016 | ||
(600mg Deleobuvir and 120mg Faldaprevir) | sgohilodlv = fbauujxyui gnawauegrc (vakqetqgkx, lfpvpghvwq - ecleflruux) View more | ||||||
Phase 1 | - | 18 | atqtyujnax(lbfzhqfbif) = rwywjamzrt yeprlxtvmj (nkhtoamsun, iisxfqqthx - tnxqjxvnlm) View more | - | 11 Apr 2016 | ||
Phase 1 | 4 | dhkdrwcmmf = lgwmnbsozp hdzlegxull (csbwhbydsl, vbjmkeszzk - cyzdcpgwit) View more | - | 11 Apr 2016 | |||
Phase 1 | - | 32 | (400 mg Deleobuvir) | eqsbslrcil = neimetloqq sfbesipiyu (mgsddmkhbl, ydekokwgkw - yeksyodjab) View more | - | 08 Apr 2016 | |
(600 mg Deleobuvir) | eqsbslrcil = iixuwbmhtp sfbesipiyu (mgsddmkhbl, swxxatolzu - louojpdius) View more |