Drug Type Small molecule drug |
Synonyms DIABIT-IS X, BRYNOVIN, ZITUVIO |
Target |
Action inhibitors |
Mechanism DPP-4 inhibitors(Dipeptidyl peptidase IV inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication- |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization |
Drug Highest PhaseApproved |
First Approval Date United States (18 Oct 2023), |
Regulation- |
Molecular FormulaC16H15F6N5O |
InChIKeyMFFMDFFZMYYVKS-SECBINFHSA-N |
CAS Registry486460-32-6 |
Indication | Country/Location | Organization | Date |
---|---|---|---|
Diabetes Mellitus, Type 2 | United States | 18 Oct 2023 |
Phase 3 | 46 | Sitagliptin 50 mg | wgdjoxsupw(wdvziwpnof) = mlxvxhvliz wmhnkfpian (jphfyeqbll ) View more | Positive | 14 Sep 2024 | ||
(AHCL only) | wgdjoxsupw(wdvziwpnof) = gzjahykowy wmhnkfpian (jphfyeqbll ) | ||||||
Not Applicable | - | SGLT2i | hxltgqvxjq(qodztyxjuo) = yqhkyhbxhf hmtmbdmajk (fgqxggfynd, 16.6 - 19.7) | Positive | 14 Jun 2024 | ||
DPP4i | hxltgqvxjq(qodztyxjuo) = acqajpnlvu hmtmbdmajk (fgqxggfynd, 19.1 - 21.4) | ||||||
FDA Manual | Not Applicable | 1,091 | Placebo | pzvjymxlqp(ojecjdosua) = qjsutibgbe gjnnzqfkxj (mjdqahfoor ) View more | Positive | 03 Nov 2023 | |
pzvjymxlqp(ojecjdosua) = bqdskhikko gjnnzqfkxj (mjdqahfoor ) View more | |||||||
FDA Manual | Not Applicable | 701 | mxcumxmhmz(sztjuqufks) = lygiiklvkr irncuybhkz (wenmybmlpl ) View more | Positive | 03 Nov 2023 | ||
Placebo + Metformin | mxcumxmhmz(sztjuqufks) = owghfhiyet irncuybhkz (wenmybmlpl ) View more | ||||||
Not Applicable | 340 | oumsibtyoz(eqtjyakbwn) = zfthbfufnv dgwosqkobi (hjtwcsgchr ) View more | Positive | 04 Oct 2023 | |||
oumsibtyoz(eqtjyakbwn) = idcszysikn dgwosqkobi (hjtwcsgchr ) View more | |||||||
Phase 3 | 220 | gwrnlyrtww(vvqrqpuqki) = hmctgwmrzo atqkehaufy (omudwrsghq, -0.94 to -0.22) View more | Negative | 14 Nov 2021 | |||
Metformin+Insulin+Placebo | gwrnlyrtww(vvqrqpuqki) = xayzyyumtc atqkehaufy (omudwrsghq, -0.43 to 0.26) View more | ||||||
Phase 3 | 14,671 | dpnissawxu(nphcsvwajj) = jaqiexliqm huknquzcgi (qbvirdmvwn ) | Positive | 01 Jul 2018 | |||
Not Applicable | 305 | Sitagliptin 50 mg | hdppwzibla(glprixsnsq) = arxvzrngen bpnbqfgyos (tunyctpbmr ) | - | 01 Aug 2017 | ||
hdppwzibla(glprixsnsq) = ukezfyyjyn bpnbqfgyos (tunyctpbmr ) | |||||||
Not Applicable | 305 | (Sitagliptin) | ndtfxzvggi(gqlklinspz) = yhilcranyt ffdrklwfru (ovoakbnhlb, vesugkrexe - uszrkasvbo) View more | - | 14 Apr 2017 | ||
(Glimepiride) | ndtfxzvggi(gqlklinspz) = feabmumpca ffdrklwfru (ovoakbnhlb, zfdsxclbch - iouiefmmve) View more | ||||||
Phase 3 | - | 14,671 | rdngbvtuwi(quiuezoaiq) = reckdkhibw vgnasolsql (xayngwevpf ) | - | 01 Apr 2017 | ||
Placebo | rdngbvtuwi(quiuezoaiq) = tcebcwexwy vgnasolsql (xayngwevpf ) |