Drug Type Small molecule drug |
Synonyms OZ-439 |
Target- |
Mechanism- |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
Drug Highest PhasePhase 3 |
First Approval Date- |
Regulation- |
Molecular FormulaC28H39NO5 |
InChIKeyXLCNVWUKICLURR-VFXIDCLRSA-N |
CAS Registry1029939-86-3 |
KEGG | Wiki | ATC | Drug Bank |
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- | - | - |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Malaria, Falciparum | Phase 3 | BJ | 01 Jul 2014 | |
Malaria, Falciparum | Phase 3 | BF | 01 Jul 2014 | |
Malaria, Falciparum | Phase 3 | GA | 01 Jul 2014 | |
Malaria, Falciparum | Phase 3 | MZ | 01 Jul 2014 | |
Malaria, Falciparum | Phase 3 | CG | 01 Jul 2014 | |
Malaria, Falciparum | Phase 3 | UG | 01 Jul 2014 | |
Malaria, Falciparum | Phase 3 | VN | 01 Jul 2014 | |
Malaria | Phase 3 | - | - | |
Malaria, Vivax | Phase 2 | - | 01 Oct 2010 |
Phase 1 | 24 | (Cohort 1:Treatment Group B: 200mg of OZ439 and 640 mg PQP) | xrixbbbino(lfcsbymymt) = knxnncjurc bnknnquwmo (kqkcynhqqw, vgupybvttw - eqoakmbewt) View more | - | 10 May 2024 | ||
(Cohort 1: Treatment Group A: 200mg of OZ439 and 480 mg PQP) | xrixbbbino(lfcsbymymt) = uryhgfrjmj bnknnquwmo (kqkcynhqqw, sbgmwfgkex - zujztopxoa) View more | ||||||
Phase 1/2 | - | paqwqqcpxc(xxncdzshlj) = foqxodupvc bgafazmzkw (iufztvbjrp ) | - | 28 Jun 2021 | |||
Phase 2 | 140 | (Ferroquine 400 mg + Artefenomel 300 mg) | iyygprjvay(dqpmuleobk) = twqkfjkect pyobgqjkoz (dentuwpjja, dulimrwiqf - fauwkbdxkn) View more | - | 02 Dec 2020 | ||
(Ferroquine 400 mg + Artefenomel 600 mg) | iyygprjvay(dqpmuleobk) = xnxbfgfrzq pyobgqjkoz (dentuwpjja, lrfgmfkgdw - sstvzsudpt) View more | ||||||
Phase 2 | 377 | (Ferroquine (up to 400 mg) + Artefenomel (up to 800 mg)) | zjofkfwquj(coqlihgkrh) = ssdztuundd zzmoluswyb (duokgtjpso, savrjiwgsr - nkqwjxqxhz) View more | - | 19 Oct 2020 | ||
(Ferroquine (up to 600 mg) + Artefenomel (up to 800 mg)) | zjofkfwquj(coqlihgkrh) = ysqcmnnvxi zzmoluswyb (duokgtjpso, xgyvwxcbeo - sxmfovnckd) View more | ||||||
Phase 1/2 | 16 | (DSM265 P. Falciparum) | yizvjamvbq(sdhyasuhns) = nakcnorqui nqwlywbaiw (zvvbrfmjgl, uadadegeda - vhvgtunlwc) View more | - | 05 Jun 2020 | ||
(OZ439 P. Vivax) | yizvjamvbq(sdhyasuhns) = qebtghqgxj nqwlywbaiw (zvvbrfmjgl, rhrknzvbqw - fhgefswqpn) View more | ||||||
Phase 1/2 | 8 | lrtdzutype(skoznyydiz) = xiauupxmov gwapnsgmzu (wjitoeankb ) View more | Positive | 01 Jun 2020 | |||
Phase 1/2 | 11 | (Primaquine 15mg) | aacbpaiagq(pankdyeqtz) = svqboftdlx emovmzlaot (ygxbndghhn, dqmbmeodhp - mzllikxvwp) View more | - | 26 May 2020 | ||
(OZ439 500mg) | aacbpaiagq(pankdyeqtz) = zgkslinerp emovmzlaot (ygxbndghhn, nzkhholwms - sudeebkgsi) View more | ||||||
NCT02389348 (Pubmed) Manual | Phase 1/2 | 13 | (Cohort 1) | nacipehwbl(vhkkzcqtox) = wrvovuigei xnvedxhica (gmalmwgwfy ) View more | Positive | 20 Dec 2019 | |
(Cohort 2) | nacipehwbl(vhkkzcqtox) = bdrepoygly xnvedxhica (gmalmwgwfy ) View more | ||||||
Phase 2 | 448 | Artefenomel 800 mg + PQP 640 mg | zxvfrwuskk(xmydiekbrl) = aewsbmzgin qygccghusj (tcjaadvwdu, 61.13 - 79.19) | - | 09 Oct 2017 | ||
Artefenomel 800 mg + PQP 960 mg | zxvfrwuskk(xmydiekbrl) = vltkqdfkpx qygccghusj (tcjaadvwdu, 59.13 - 76.66) | ||||||
Phase 2 | 25 | (OZ439 100mg) | qrgwgfgdmz(kgbcarknix) = ovpmhhnfnd gqgoxfkjru (coqqznmshf, szlyisgxry - wdkahxtrqr) View more | - | 10 Feb 2017 | ||
(OZ439 500mg) | qrgwgfgdmz(kgbcarknix) = eohmxchtgo gqgoxfkjru (coqqznmshf, ophiagegau - venqcuancz) View more |