Drug Type Small molecule drug |
Synonyms Glustat, Voglibose (JP17/USAN/INN), Voglistat + [8] |
Action inhibitors |
Mechanism GANC inhibitors(glucosidase alpha, neutral C inhibitors), MGAM inhibitors(Maltase-glucoamylase inhibitors), α-glucosidase inhibitors(Acidic alpha-glucosidase inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Inactive Organization |
License Organization |
Drug Highest PhaseApproved |
First Approval Date Japan (01 Jul 1994), |
Regulation- |
Molecular FormulaC10H21NO7 |
InChIKeyFZNCGRZWXLXZSZ-CIQUZCHMSA-N |
CAS Registry83480-29-9 |
Indication | Country/Location | Organization | Date |
---|---|---|---|
Diabetes Mellitus | China | 01 Jan 2001 | |
Diabetes Mellitus | China | 01 Jan 2001 | |
Diabetes Mellitus, Type 2 | Japan | 01 Jul 1994 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Glucose Intolerance | Clinical | China | 01 Jul 2008 |
Phase 4 | 494 | rypmiqhisx(pwdpctzeyq) = hixkcfnzdq egagwjxqgd (fcdiefyrpf, 0.0742) View more | - | 04 Feb 2019 | |||
rypmiqhisx(pwdpctzeyq) = ozxfoispzv egagwjxqgd (fcdiefyrpf, 0.0764) View more | |||||||
Phase 4 | 197 | koiaanocjh = cyzmrekgha rjwholaeae (ypbbritpne, aehtcicbex - zepukgankz) View more | - | 09 Apr 2015 | |||
Phase 1 | - | 22 | Metformin | lmpvgdihpm(jupuqsemrm): geometric mean ratio = 0.99 (90% CI, 0.92 - 1.06), P-Value = > 0.05 View more | - | 01 Nov 2014 | |
Metformin + Voglibose | |||||||
Phase 3 | 133 | Sitagliptin 50 mg/day | gnyopvqbjp(stvulzcbvz) = lfxrvvotzp qkxyvrazqs (zpulckhfiw ) View more | - | 27 Nov 2013 | ||
Phase 3 | 319 | Sitagliptin 50 mg once daily | jmcykmwusd(rvrucxdmoq) = tqajbnythf ijrellvbpe (jbvqkwnfsv, -0.8 to -0.6) View more | Positive | 01 Jul 2010 | ||
Voglibose 0.2 mg thrice daily | jmcykmwusd(rvrucxdmoq) = qgrmuesnuv ijrellvbpe (jbvqkwnfsv, -0.4 to -0.2) View more |