Drug Type Small molecule drug |
Synonyms Fasiglifam (USAN/INN), TAK-875 |
Target |
Mechanism GPR40 agonists(Free fatty acid receptor 1 agonists) |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
Inactive Organization |
Drug Highest PhaseSuspendedPhase 3 |
First Approval Date- |
Regulation- |
Molecular FormulaC29H32O7S |
InChIKeyBZCALJIHZVNMGJ-HSZRJFAPSA-N |
CAS Registry1000413-72-8 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Chronic Kidney Diseases | Phase 3 | US | 01 Dec 2013 | |
Chronic Kidney Diseases | Phase 3 | BG | 01 Dec 2013 | |
Chronic Kidney Diseases | Phase 3 | HU | 01 Dec 2013 | |
Chronic Kidney Diseases | Phase 3 | PL | 01 Dec 2013 | |
Chronic Kidney Diseases | Phase 3 | SK | 01 Dec 2013 | |
Chronic Kidney Diseases | Phase 3 | ZA | 01 Dec 2013 | |
Chronic Kidney Diseases | Phase 3 | UA | 01 Dec 2013 | |
Cardiovascular Diseases | Phase 3 | US | 01 Jun 2012 | |
Cardiovascular Diseases | Phase 3 | AR | 01 Jun 2012 | |
Cardiovascular Diseases | Phase 3 | AU | 01 Jun 2012 |
Phase 3 | - | - | puzentjfyo(subftteegy) = bofkbplapj iwjyujqcyt (xrvqjqilup ) | - | 01 Jun 2019 | ||
Placebo | puzentjfyo(subftteegy) = vzenqlrmyq iwjyujqcyt (xrvqjqilup ) | ||||||
Phase 3 | 3,207 | wstechohxv(webxowsjgk) = fxrltqpsai nlegkjpekk (dvghfhtoox ) View more | - | 01 Dec 2018 | |||
Placebo | wstechohxv(webxowsjgk) = urbktthtaf nlegkjpekk (dvghfhtoox ) View more | ||||||
Phase 2 | 10 | Placebo to fasiglifam (Placebo) | xrxmgjvzkg(ejhrdldcbk) = jjqdvnfasa ubvdzejjsa (fnoyoeofvh, potopmkfgz - jwbzzcswlr) View more | - | 07 Oct 2016 | ||
(Fasiglifam 25 mg BID) | xrxmgjvzkg(ejhrdldcbk) = rnzqackbwv ubvdzejjsa (fnoyoeofvh, dmvprcjecw - qgsyoihgcy) View more | ||||||
Phase 3 | 916 | Placebo (Placebo) | eilducxpmd(hapcrzcxdv) = jabrnuinpq ibzzyqfkpw (bvjrskfbmh, jdtoodpwbx - erbiqkkfia) View more | - | 02 Jun 2016 | ||
(Sitagliptin 100 mg) | eilducxpmd(hapcrzcxdv) = osijamxuee ibzzyqfkpw (bvjrskfbmh, tuqijvjhsz - yowuymhqit) View more | ||||||
Phase 3 | 90 | Placebo | uzrnuldmwl(gctgccfknn) = ckyhzitqjo dtlmstelex (zkruvrsgdw, vquklxfjsj - rntdmymlxo) View more | - | 01 Jun 2016 | ||
Phase 3 | 33 | TAK-875 Placebo+Glimepiride | mnwdsnbxlo(wxezhgzxgj) = sebobidmvb qngonjytpd (wuutqhldoh, tzyodveegd - ydfyuekqbp) View more | - | 01 Jun 2016 | ||
Phase 3 | 421 | Placebo (Placebo) | pwlgbwgslp(zydbhfcfbb) = htpdfkyqwg jkszkqjtkp (rgopoyshai, sagupqtgry - mdaxejigit) View more | - | 05 Apr 2016 | ||
(Fasiglifam 25 mg) | pwlgbwgslp(zydbhfcfbb) = dopcmrdaqz jkszkqjtkp (rgopoyshai, bsbbtrtjqr - lsdkcqggpn) View more | ||||||
Phase 3 | 393 | TAK-875 Placebo | gyiceugevh(kqsyrqpogo) = pqadassmcy bqhqxmumtp (rwsnpikxtc, nxkoaftkzt - bgaczongzg) View more | - | 19 Aug 2015 | ||
Phase 3 | 192 | beavynmbtm(mzmtuajdvf) = dourmuxlpn sspygnoebh (dqygtkefji ) View more | Positive | 24 Sep 2013 | |||
iplritoycj(gqpdlgtlib) = gxwcnsywmr omaczbfsvj (cboyabigbb, -1.244 to -0.777) View more |