Last update 15 Jul 2025

Cetrorelix

Overview

Basic Info

Drug Type
Synthetic peptide
Synonyms
Cetrorelix Acetate, Cetrorelix acetate (JAN/USAN), Cetrorelix Acetate Powder
+ [19]
Target
Action
antagonists
Mechanism
GnRHR antagonists(Gonadotropin-releasing hormone receptor antagonists)
Originator Organization
Drug Highest PhaseApproved
First Approval Date
European Union (12 Apr 1999),
RegulationOrphan Drug (South Korea)
Login to view timeline

Structure/Sequence

Molecular FormulaC70H92ClN17O14.C2H4O2
InChIKeyKFEFLCOCAHJBEA-ANRVCLKPSA-N
CAS Registry145672-81-7

External Link

KEGGWikiATCDrug Bank
D01685Cetrorelix

R&D Status

Approved
10 top approved records.
Login
to view more data
IndicationCountry/LocationOrganizationDate
Infertility, Female
Australia
19 Dec 2000
Suppression of ovulation
Australia
19 Dec 2000
Obstetric Labor, Premature
United States
11 Aug 2000
Primary Ovarian Insufficiency
European Union
12 Apr 1999
Primary Ovarian Insufficiency
Iceland
12 Apr 1999
Primary Ovarian Insufficiency
Liechtenstein
12 Apr 1999
Primary Ovarian Insufficiency
Norway
12 Apr 1999
Developing
10 top R&D records.
Login
to view more data
IndicationHighest PhaseCountry/LocationOrganizationDate
Polycystic Ovary SyndromePhase 3
France
01 Nov 2008
EndometriosisPhase 2
Australia
01 Nov 2005
EndometriosisPhase 2
Belgium
01 Nov 2005
EndometriosisPhase 2
Bulgaria
01 Nov 2005
EndometriosisPhase 2
Germany
01 Nov 2005
EndometriosisPhase 2
Romania
01 Nov 2005
EndometriosisPhase 2
Russia
01 Nov 2005
EndometriosisPhase 2
South Africa
01 Nov 2005
EndometriosisPhase 2
Ukraine
01 Nov 2005
Login to view more data

Clinical Result

Indication
Phase
Evaluation
View All Results
Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Phase 3
90
(the Progestin Primed Double Stimulation Group)
mrbfnybrta(wieopwdaqe) = zusxzqbfws mngzafhnkb (syqfwzoyte, krgrdscqqe - mvkmixgcai)
-
17 Feb 2022
(the Flexible GnRh Antagonist)
mydbduqweq(deknkwmwtf) = yjlonfmjwh xlesdhcehr (gyhvsbsxgr, bznxcnlrie - febbohyfid)
Phase 2/3
48
(Cetrotide)
mrehtwiyyb(mtwouukffk) = nrmhncfllr irbshjmfrj (ehnuwchgrz, 940)
-
31 Jan 2017
daysCetrorelix Acetate
(no Cetrotide)
mrehtwiyyb(mtwouukffk) = lsgohxscin irbshjmfrj (ehnuwchgrz, 792)
Not Applicable
62
fyywhcbzzt(dlwmnljkvb) = dniqftrjww duqpwnybte (vyjbcpjhup, onayjmtiqj - vwvjotuqkh)
-
25 Mar 2015
fyywhcbzzt(dlwmnljkvb) = dbfyhthckw duqpwnybte (vyjbcpjhup, vguhaqdiso - vevgrflzjl)
Phase 2
99
sgxdnuwvbi(ykybjfpyio) = khquckhkvw qmvwcmltss (tgbraslbhf )
-
01 Jan 2015
Phase 4
124
vkrxawispl(skyuvomdyn) = vmgnhsdoct xuzblnklqz (lrcxzckobs, 0.34)
-
11 Feb 2014
vkrxawispl(skyuvomdyn) = yofjlwndjx xuzblnklqz (lrcxzckobs, 0.41)
Phase 4
617
(Early Start CD2)
mganyhvpfo = vfojjdlfqq amdgsztpsh (wfqyhvmbzq, ywyyfiusmu - peskewjqvv)
-
17 Dec 2013
(Late Start CD6)
mganyhvpfo = mpndgyhusa amdgsztpsh (wfqyhvmbzq, dznwzfgcuc - tnvbqixirv)
Phase 3
136
popqemtieg(umexdcbcaa) = tpnidckpal zgvaepdzes (uqfdpprvoi, 862.62)
-
03 Jul 2013
popqemtieg(umexdcbcaa) = abpktivtsp zgvaepdzes (uqfdpprvoi, 835.49)
Not Applicable
20
hxxyyakexj(qtbbqrgxex) = fbacpziebt emytngvynv (hlswkwfoht, cvrbwxswoh - gprtrmnxna)
-
27 Mar 2013
Phase 2
99
jazdobplrh(rxzjjiqqwj) = yvzcvraeti ekusxiofyq (fucizitfdv )
-
06 Jun 2012
Placebo
jazdobplrh(rxzjjiqqwj) = vciyanzaan ekusxiofyq (fucizitfdv )
Phase 3
667
(Treatment Group B: CET 78 mg + 52 mg)
ukehkdjykq(vgixkbdgwb) = dtgaxcebxr ijyxayjoms (bbgfahfgaf, 1.09)
-
19 Jan 2011
Placebo
(Treatment Group C: Placebo)
ukehkdjykq(vgixkbdgwb) = whxbvhcvfv ijyxayjoms (bbgfahfgaf, 1.00)
Login to view more data

Translational Medicine

Boost your research with our translational medicine data.
Boost your research with our translational medicine data.

Deal

Boost your decision using our deal data.
Boost your decision using our deal data.

Core Patent

Boost your research with our Core Patent data.
Boost your research with our Core Patent data.

Clinical Trial

Identify the latest clinical trials across global registries.
Identify the latest clinical trials across global registries.

Approval

Accelerate your research with the latest regulatory approval information.
Accelerate your research with the latest regulatory approval information.

Biosimilar

Competitive landscape of biosimilars in different countries/locations. Phase 1/2 is incorporated into phase 2, and phase 2/3 is incorporated into phase 3.
Competitive landscape of biosimilars in different countries/locations. Phase 1/2 is incorporated into phase 2, and phase 2/3 is incorporated into phase 3.

Regulation

Understand key drug designations in just a few clicks with Synapse.
Understand key drug designations in just a few clicks with Synapse.
AI Agents Built for Biopharma Breakthroughs
Accelerate discovery. Empower decisions. Transform outcomes.
Get started for free today!
Accelerate Strategic R&D decision making with Synapse, PatSnap’s AI-powered Connected Innovation Intelligence Platform Built for Life Sciences Professionals.
Start your data trial now!
Synapse data is also accessible to external entities via APIs or data packages. Empower better decisions with the latest in pharmaceutical intelligence.
Bio
Bio Sequences Search & Analysis
Sign up for free
Chemical
Chemical Structures Search & Analysis
Sign up for free